SCHEMBL8276293

SCHEMBL8276293

COc1ccc2c(O[C@@H]3CC(C(N)=O)N(C(=O)[C@@H](NC(=O)OC4CCCC4)C(C)(C)C)C3)cc(-c3csc(NC(C)C)n3)nc2c1

nearest known ligand 0.74

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CTSB P07858 1/20 0.53
PPP3CB P16298 1/20 0.53
ABCC1 P33527 1/20 0.48
ABCC2 Q92887 1/20 0.48
ABCG2 Q9UNQ0 1/20 0.48
ADRB3 P13945 1/20 0.40
ADRA2B P18089 1/20 0.40
ADRA2C P18825 1/20 0.40
CYP3A4 P08684 2/20 0.37
ELANE P08246 1/20 0.32
P2RX3 P56373 1/20 0.32
KCNQ1 P51787 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8274031 1.00 CTSB (0.53) CTSBPPP3CBABCC1ABCC2ABCG2
SCHEMBL13522781 0.94 CTSB (0.55) CTSBPPP3CBABCC1ABCC2ABCG2
SCHEMBL8274106 0.94 CTSB (0.55) CTSBPPP3CBABCC1ABCC2ABCG2
SCHEMBL8272992 0.94 CTSB (0.55) CTSBPPP3CBABCC1ABCC2ABCG2
SCHEMBL10193686 0.94 CTSB (0.54) CTSBPPP3CBABCC1ABCC2ABCG2
SCHEMBL693682 0.94 CTSB (0.55) CTSBPPP3CBABCC1ABCC2ABCG2
SCHEMBL8273160 0.94 CTSB (0.60) CTSBPPP3CBABCC1ABCC2ABCG2
SCHEMBL12676434 0.93 CTSB (0.52) CTSBPPP3CBABCC1ABCC2ABCG2
SCHEMBL8273175 0.91 CTSB (0.49) CTSBPPP3CBABCC1ABCC2ABCG2
SCHEMBL8273042 0.89 CTSB (0.48) CTSBPPP3CBABCC1ABCC2ABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006020276-A2 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. (US) 2006-02-23 WO disclosed