SCHEMBL8280378

SCHEMBL8280378

COc1cnn(C)c(=O)c1-c1ccc(C[C@H](NC(=O)C(C(C)C)n2c(C)cc(C(=O)c3ccccc3)c2C)C(=O)O)cc1

nearest known ligand 0.61

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 20/20 0.61
ITGB7 P26010 20/20 0.61
ITGB1 P05556 9/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6029076 1.00 ITGA4 (0.61) ITGA4ITGB7ITGB1
SCHEMBL8280377 0.95 ITGA4 (0.54) ITGA4ITGB7ITGB1
SCHEMBL8282667 0.88 ITGA4 (0.72) ITGA4ITGB7ITGB1
SCHEMBL6030313 0.88 ITGA4 (0.72) ITGA4ITGB7ITGB1
SCHEMBL6029072 0.82 ITGA4 (0.43) ITGA4ITGB7ITGB1
SCHEMBL8282990 0.82 ITGA4 (0.71) ITGA4ITGB7ITGB1
SCHEMBL6028815 0.82 ITGA4 (0.71) ITGA4ITGB7ITGB1
SCHEMBL8280376 0.81 ITGA4 (0.61) ITGA4ITGB7ITGB1
SCHEMBL6029683 0.79 ITGA4 (0.76) ITGA4ITGB7ITGB1
SCHEMBL8281604 0.79 ITGA4 (0.76) ITGA4ITGB7ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005077915-A1 PYRIDAZINONES AS ANTAGONISTS OF A4 INTEGRINS JANSSEN PHARMACEUTICA, N.V. (BE) 2005-08-25 WO disclosed