SCHEMBL8280939

SCHEMBL8280939

COC[C@H](C)Oc1ccc(-c2nnc(CO)o2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.50
NOTUM Q6P988 1/20 0.50
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 3/20 0.46
HPGD P15428 3/20 0.46
POLB P06746 1/20 0.46
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
HDAC8 Q9BY41 2/20 0.46
RAB9A P51151 5/20 0.42
NPC1 O15118 4/20 0.42
TSHR P16473 2/20 0.42
HSD17B10 Q99714 2/20 0.42
LMNA P02545 1/20 0.42
SMPD1 P17405 1/20 0.42
NR1H4 Q96RI1 1/20 0.41
PRKAB2 O43741 2/20 0.41
PRKAG1 P54619 2/20 0.41
PRKAA2 P54646 2/20 0.41
PRKAA1 Q13131 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8281642 1.00 MAPT (0.50) MAPTNOTUMKDM4EALDH1A1HPGD
SCHEMBL8280935 0.85 MAPT (0.48) MAPTKDM4EALDH1A1HPGDPOLB
SCHEMBL8282545 0.84 MAPT (0.47) MAPTKDM4EALDH1A1HPGDPOLB
SCHEMBL8280938 0.83 MAPT (0.49) MAPTKDM4EALDH1A1HPGDPOLB
SCHEMBL97043 0.72 NOTUM (0.68) MAPTNOTUMKDM4EALDH1A1HPGD
SCHEMBL5637347 0.71 LSS (0.51) MAPTNOTUMKDM4EALDH1A1HPGD
SCHEMBL14409749 0.70 ESR2 (0.52) MAPTALDH1A1HPGDPOLBCYP2C9
SCHEMBL95172 0.70 NOTUM (0.60) MAPTNOTUMKDM4EALDH1A1HPGD
SCHEMBL1270235 0.69 GCK (0.52) NR1H4
SCHEMBL9898682 0.69 GCK (0.52) NR1H4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082866-A2 SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-09-09 WO disclosed