SCHEMBL8280935

SCHEMBL8280935

COC[C@@H](C)Oc1ccc(-c2nnc(COC(C)C)o2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 6/20 0.48
ALDH1A1 P00352 5/20 0.44
POLB P06746 5/20 0.44
KDM4E B2RXH2 4/20 0.44
HPGD P15428 4/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
HDAC8 Q9BY41 2/20 0.41
RAB9A P51151 6/20 0.41
NPC1 O15118 5/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
TSHR P16473 3/20 0.40
HSD17B10 Q99714 3/20 0.40
LMNA P02545 2/20 0.40
TP53 P04637 1/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.38
MAPK1 P28482 1/20 0.38
SMPD1 P17405 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8282545 0.86 MAPT (0.47) MAPTALDH1A1POLBKDM4EHPGD
SCHEMBL8281642 0.85 MAPT (0.50) MAPTALDH1A1POLBKDM4EHPGD
SCHEMBL8280939 0.85 MAPT (0.50) MAPTALDH1A1POLBKDM4EHPGD
SCHEMBL8280938 0.81 MAPT (0.49) MAPTALDH1A1POLBKDM4EHPGD
SCHEMBL2088807 0.72 MAPT (0.69) MAPTALDH1A1POLBKDM4EHPGD
SCHEMBL14409749 0.69 ESR2 (0.52) MAPTALDH1A1POLBHPGDCYP2C9
SCHEMBL2090020 0.68 NPC1 (0.57) MAPTALDH1A1POLBKDM4EHPGD
SCHEMBL2093543 0.67 NPSR1 (0.52) MAPTALDH1A1POLBKDM4EHPGD
SCHEMBL6530672 0.67 S1PR1 (0.47) MAPTALDH1A1POLBKDM4EHPGD
SCHEMBL9406398 0.66 LTA4H (0.42) KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082866-A2 SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-09-09 WO disclosed