SCHEMBL8282104

SCHEMBL8282104

COc1cnn(C)c(=O)c1-c1ccc(C[C@H](NC(=O)OC(C)(C)C)C(=O)O)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 20/20 1.00
ITGB7 P26010 20/20 1.00
ITGB1 P05556 9/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8282103 0.93 ITGA4 (0.86) ITGA4ITGB7ITGB1
SCHEMBL8282997 0.92 ITGA4 (0.84) ITGA4ITGB7ITGB1
SCHEMBL6469692 0.92 ITGA4 (0.84) ITGA4ITGB7ITGB1
SCHEMBL24946013 0.91 ITGA4 (1.00) ITGA4ITGB7ITGB1
SCHEMBL24946012 0.91 ITGA4 (0.83) ITGA4ITGB7ITGB1
SCHEMBL24945961 0.89 ITGA4 (1.00) ITGA4ITGB7ITGB1
SCHEMBL6028867 0.85 ITGA4 (1.00) ITGA4ITGB7ITGB1
SCHEMBL8282992 0.85 ITGA4 (0.74) ITGA4ITGB7ITGB1
SCHEMBL6028861 0.85 ITGA4 (1.00) ITGA4ITGB7ITGB1
SCHEMBL24945903 0.85 ITGA4 (1.00) ITGA4ITGB7ITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005077915-A1 PYRIDAZINONES AS ANTAGONISTS OF A4 INTEGRINS JANSSEN PHARMACEUTICA, N.V. (BE) 2005-08-25 WO disclosed
WO-2005077914-A1 PYRIDAZINONE UREAS AS ANTAGONISTS OF α4 INTEGRINS JANSSEN PHARMACEUTICA, N.V. (BE) 2005-08-25 WO disclosed