SCHEMBL8284682

SCHEMBL8284682

CCOC(=O)c1nc(-c2ccccc2Cl)n(-c2ccc(Cl)cc2)c1/C=N/N

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 13/20 0.47
CHRNA7 P36544 1/20 0.45
CNR2 P34972 7/20 0.45
KDM4E B2RXH2 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
GABRA2 P47869 3/20 0.41
GABRB2 P47870 3/20 0.41
MAPK1 P28482 1/20 0.41
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5370296 1.00 CNR1 (0.47) CNR1CHRNA7CNR2KDM4ENPC1
SCHEMBL5370292 1.00 CNR1 (0.47) CNR1CHRNA7CNR2KDM4ENPC1
SCHEMBL5339713 0.88 CNR1 (0.50) CNR1CHRNA7CNR2KDM4ENPC1
SCHEMBL6332827 0.83 CNR1 (0.53) CNR1CHRNA7CNR2KDM4ENPC1
SCHEMBL5350855 0.81 CNR1 (0.56) CNR1CHRNA7CNR2KDM4ENPC1
SCHEMBL739526 0.81 CNR1 (0.64) CNR1CNR2KDM4ENPC1RAB9A
SCHEMBL4277527 0.80 CNR1 (0.55) CNR1CHRNA7CNR2KDM4ENPC1
SCHEMBL6357570 0.78 CNR1 (0.57) CNR1CNR2KDM4E
SCHEMBL6360811 0.76 CNR1 (0.55) CNR1CNR2KDM4ENPC1RAB9A
SCHEMBL1040785 0.73 CNR1 (0.74) CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070213334-A1 CANNABINOID RECEPTOR LIGANDS AND USES THEREOF CARPINO PHILIP A 2007-09-13 US disclosed
US-20070213334-A1 CANNABINOID RECEPTOR LIGANDS AND USES THEREOF CARPINO PHILIP A 2007-09-13 US disclosed
US-7232823-B2 Cannabinoid receptor ligands and uses thereof PFIZER, INC. (US) 2007-06-19 US disclosed
US-7232823-B2 Cannabinoid receptor ligands and uses thereof PFIZER, INC. (US) 2007-06-19 US disclosed
WO-2005061504-A1 BICYCLIC PYRIDAZINONE CANNABINOID RECEPTOR LIGANDS AND USES THEREOF PFIZER PRODUCTS INC. (US) 2005-07-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070213334-A1 CANNABINOID RECEPTOR LIGANDS AND USES THEREOF CNR2, CNR1, GPR18 CNR1 2/4885CHRNA7 142/4885CNR2 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.