SCHEMBL8285409

SCHEMBL8285409

O=C(N[C@H](C(=O)O)C1CCCCC1)c1ccccn1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.53
EGFR P00533 1/20 0.53
ERBB2 P04626 1/20 0.53
MET P08581 1/20 0.53
KDR P35968 1/20 0.53
MERTK Q12866 1/20 0.53
GRM4 Q14833 2/20 0.52
GAA P10253 3/20 0.51
CYP1A2 P05177 1/20 0.51
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 1/20 0.50
KDM4E B2RXH2 1/20 0.50
PYGL P06737 4/20 0.48
MMP13 P45452 1/20 0.47
EPHX2 P34913 2/20 0.46
FPR2 P25090 1/20 0.46
MAPT P10636 2/20 0.46
PKM P14618 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8285399 0.86 ALDH1A1 (0.50) GRM5EGFRERBB2METKDR
SCHEMBL7857535 0.81 MAPT (0.54) GAACYP1A2NPC1RAB9ASMN1; SMN2
SCHEMBL329840 0.81 MAPT (0.54) GAACYP1A2NPC1RAB9ASMN1; SMN2
SCHEMBL14087347 0.81 GRM5 (0.52) GRM5EGFRERBB2METKDR
SCHEMBL21274424 0.78 CCR1 (0.56) NPC1RAB9AALDH1A1PYGL
SCHEMBL21274426 0.78 CCR1 (0.56) NPC1RAB9AALDH1A1PYGL
SCHEMBL4000977 0.77 GRM5 (0.62) GRM5EGFRERBB2METKDR
SCHEMBL3210060 0.77 MAPT (0.50) GAASMN1; SMN2ALDH1A1FPR2MAPT
SCHEMBL3210085 0.77 MAPT (0.50) GAASMN1; SMN2ALDH1A1FPR2MAPT
SCHEMBL22449377 0.77 GRM5 (0.80) GRM5EGFRERBB2METKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7485625-B2 Inhibitors of hepatitis C virus NS3/NS4a serine protease SCHERING CORPORATION (US) 2009-02-03 US disclosed
US-7485625-B2 Inhibitors of hepatitis C virus NS3/NS4a serine protease SCHERING CORPORATION (US) 2009-02-03 US disclosed
WO-2005058821-A1 INHIBITORS OF HEPATITIS C VIRUS NS3/NS4A SERINE PROTEASE SCHERING CORPORATION (US) 2005-06-30 WO disclosed