SCHEMBL8288683

SCHEMBL8288683

CC(C)(C)NC(=O)Nc1sc2c(c1C(N)=O)CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.57
KDM4E B2RXH2 5/20 0.53
L3MBTL1 Q9Y468 2/20 0.53
ALDH1A1 P00352 4/20 0.53
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
MAPT P10636 2/20 0.50
HPGD P15428 2/20 0.50
HSD17B10 Q99714 2/20 0.50
LMNA P02545 1/20 0.50
TP53 P04637 1/20 0.50
ALOX15 P16050 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
POLB P06746 1/20 0.47
CASP6 P55212 1/20 0.45
KCNH2 Q12809 2/20 0.45
GAA P10253 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8288701 0.88 ADORA1 (0.55) ADORA1KDM4EL3MBTL1ALDH1A1MEN1
SCHEMBL8289859 0.85 MEN1 (0.68) ADORA1KDM4EL3MBTL1ALDH1A1MEN1
SCHEMBL8289721 0.84 ALDH1A1 (0.52) ADORA1KDM4EL3MBTL1ALDH1A1MEN1
SCHEMBL351566 0.84 KCNH2 (0.66) ADORA1KDM4EALDH1A1MEN1KMT2A
SCHEMBL31208315 0.81 ADORA1 (0.48) ADORA1KDM4EL3MBTL1ALDH1A1MEN1
SCHEMBL351992 0.80 ADORA1 (0.82) ADORA1KDM4EL3MBTL1ALDH1A1MEN1
SCHEMBL16450569 0.80 KMT2A (0.54) ADORA1KDM4EALDH1A1MEN1KMT2A
SCHEMBL13738138 0.79 NPC1 (0.61) ADORA1KDM4EL3MBTL1ALDH1A1MEN1
SCHEMBL17018774 0.79 KCNH2 (0.61) KDM4EALDH1A1MEN1KMT2AMAPT
SCHEMBL13736559 0.78 ADORA1 (0.68) ADORA1KDM4EL3MBTL1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed