SCHEMBL8288774

SCHEMBL8288774

Cc1c(Br)c(C(F)(F)F)nn1CC(=O)Nc1sc2c(c1C(N)=O)CCCC2

nearest known ligand 0.66

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 16/20 0.66
GRIA2 P42262 2/20 0.61
ALDH1A1 P00352 2/20 0.56
MAPT P10636 1/20 0.56
GAA P10253 2/20 0.55
HPGD P15428 1/20 0.55
TSHR P16473 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4141384 0.99 GRM1 (0.65) GRM1GRIA2ALDH1A1MAPTGAA
SCHEMBL4152901 0.85 GRM1 (0.81) GRM1GRIA2ALDH1A1MAPTGAA
SCHEMBL3280341 0.84 ALDH1A1 (0.73) GRM1ALDH1A1MAPTGAAHPGD
SCHEMBL6861991 0.81 GRM1 (0.67) GRM1GRIA2ALDH1A1MAPTGAA
SCHEMBL29383334 0.80 HPGD (0.76) GRM1GRIA2ALDH1A1MAPTGAA
SCHEMBL1007269 0.79 GRM1 (1.00) GRM1GRIA2ALDH1A1MAPTGAA
SCHEMBL1007297 0.79 GRM1 (0.87) GRM1GRIA2ALDH1A1GAAHPGD
SCHEMBL3452590 0.79 GRM1 (0.62) GRM1GRIA2ALDH1A1MAPTGAA
SCHEMBL1007789 0.78 GRM1 (0.68) GRM1GRIA2ALDH1A1MAPTGAA
SCHEMBL1008341 0.78 GRM1 (0.71) GRM1GRIA2ALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed