SCHEMBL8289503

SCHEMBL8289503

CCCC(C)C(=O)Nc1sc2c(c1C(N)=O)CCC2

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.65
MAPK1 P28482 1/20 0.65
ALDH1A1 P00352 7/20 0.63
RAB9A P51151 7/20 0.63
SMN1; SMN2 Q16637 5/20 0.63
KMT2A Q03164 4/20 0.63
MEN1 O00255 3/20 0.63
MAPK10 P53779 1/20 0.63
FLT3 P36888 4/20 0.62
NPSR1 Q6W5P4 2/20 0.61
MAPT P10636 5/20 0.59
LMNA P02545 3/20 0.59
CYP1A2 P05177 1/20 0.59
CYP2C19 P33261 1/20 0.59
HPGD P15428 3/20 0.58
NPC1 O15118 5/20 0.58
RXFP1 Q9HBX9 1/20 0.57
TSHR P16473 2/20 0.55
ALOX15 P16050 1/20 0.55
HSD17B10 Q99714 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3912860 0.88 FLT3 (0.68) KDM4EMAPK1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL8290635 0.86 FLT3 (0.67) KDM4EMAPK1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL5467278 0.84 CFTR (0.59) KDM4EMAPK1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL8289513 0.84 KDM4E (0.70) KDM4EMAPK1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL21082573 0.82 KDM4E (0.68) KDM4EMAPK1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL20548014 0.82 KDM4E (0.68) KDM4EMAPK1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL3917266 0.82 ALDH1A1 (0.77) KDM4EMAPK1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL5459064 0.80 ALDH1A1 (0.63) KDM4EMAPK1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL8289412 0.79 KDM4E (1.00) KDM4EMAPK1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL8289831 0.79 ALDH1A1 (0.78) KDM4EMAPK1ALDH1A1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005033102-A2 THIOPHENE-BASED COMPOUNDS EXHIBITING ATP-UTILIZING ENZYME INHIBITORY ACTIVITY, AND COMPOSITIONS, AND USES THEREOF AMPHORA DISCOVERY CORPORATION (US) 2005-04-14 WO disclosed