SCHEMBL8291360

SCHEMBL8291360

C=CCOC(=O)c1cc(-c2ccc(/C=C3/C(=O)N(CCCO)C(=O)C(N)=C3C)o2)ccc1Cl

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.59
KMT2A Q03164 5/20 0.59
POLB P06746 5/20 0.59
MEN1 O00255 4/20 0.59
KDM4E B2RXH2 4/20 0.59
MAPT P10636 4/20 0.59
HPGD P15428 3/20 0.59
RECQL P46063 2/20 0.59
MCL1 Q07820 2/20 0.59
TDP1 Q9NUW8 2/20 0.59
DNMT1 P26358 1/20 0.59
BLM P54132 1/20 0.59
XPA P23025 8/20 0.59
GSK3A P49840 3/20 0.55
GSK3B P49841 3/20 0.55
ESR2 Q92731 1/20 0.52
L3MBTL1 Q9Y468 3/20 0.49
APEX1 P27695 2/20 0.48
NTSR1 P30989 1/20 0.48
GALK1 P51570 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8291312 0.89 KMT2A (0.72) ALDH1A1KMT2APOLBMEN1KDM4E
SCHEMBL8290432 0.80 ESR2 (0.72) ALDH1A1KMT2APOLBMEN1KDM4E
SCHEMBL8290360 0.79 ESR2 (0.81) ALDH1A1KMT2APOLBMEN1KDM4E
SCHEMBL19419927 0.79 ESR2 (0.69) ALDH1A1KMT2APOLBMEN1KDM4E
SCHEMBL13708915 0.78 ESR2 (0.62) ALDH1A1KMT2APOLBMEN1KDM4E
SCHEMBL19425313 0.78 ESR2 (0.62) ALDH1A1KMT2APOLBMEN1KDM4E
SCHEMBL8291279 0.78 ESR2 (0.66) ALDH1A1KMT2APOLBMEN1KDM4E
SCHEMBL14584108 0.77 ESR2 (0.62) ALDH1A1KMT2APOLBMEN1KDM4E
SCHEMBL12027509 0.76 GSK3A (0.84) ALDH1A1KMT2APOLBMEN1KDM4E
SCHEMBL8291189 0.75 POLB (0.44) ALDH1A1KMT2APOLBMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005034940-A2 DUAL ALANYL AMINOPEPTIDASE AND DIPEPTIDYL PEPTIDASE IV INHIBITORS FOR FUNCTIONALLY INFLUENCING DIFFERENT CELLS AND FOR TREATING IMMUNOLOGICAL, INFLAMMATORY, NEURONAL AND OTHER DISEASES IMTM GMBH (DE) 2005-04-21 WO disclosed