SCHEMBL8293141

SCHEMBL8293141

Cc1c(CC(=O)NN)c2cc(Cl)ccc2n1Cc1cccc(Cl)c1

nearest known ligand 0.83

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
PLA2G2A P14555 20/20 0.83

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8301132 0.93 PLA2G2A (0.78) PLA2G2A
SCHEMBL8293051 0.92 PLA2G2A (0.87) PLA2G2A
SCHEMBL8300434 0.91 PLA2G2A (1.00) PLA2G2A
SCHEMBL7953268 0.90 PLA2G2A (1.00) PLA2G2A
SCHEMBL27398701 0.87 PLA2G2A (0.70) PLA2G2A
SCHEMBL2006287 0.86 PLA2G2A (0.66) PLA2G2A
SCHEMBL8291463 0.84 PLA2G2A (0.77) PLA2G2A
SCHEMBL8292857 0.83 PLA2G2A (0.80) PLA2G2A
SCHEMBL8296288 0.83 PLA2G2A (0.64) PLA2G2A
SCHEMBL8292911 0.82 PLA2G2A (0.78) PLA2G2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1067986-C 1H-indole-3-acetic acid hydrazide spla2 inhibitors LILLY CO ELI (US) 2001-07-04 CN disclosed
EP-0620214-B1 1H-indole-3-acetic acid hydrazide sPLA2 inhibitors LILLY CO ELI (US) 1999-03-03 EP disclosed
US-5578634-A SEPTIC SHOCK TREATMENT ELI LILLY AND COMPANY (US) 1996-11-26 US disclosed
CN-1098714-A The 1H-indole-3-acetic acid hydrazide spla 2 inhibitors LILLY CO ELI (US) 1995-02-15 CN disclosed
EP-0620214-A1 1H-indole-3-acetic acid hydrazide sPLA2 inhibitors ELI LILLY AND COMPANY (US) 1994-10-19 EP disclosed