SCHEMBL8294235

SCHEMBL8294235

N[C@@H](CCCCNC(=O)c1cnc2ccccc2n1)C(=O)N1CC(F)(F)C1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.50
HDAC1 Q13547 1/20 0.50
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
HTR1A P08908 9/20 0.46
DRD2 P14416 1/20 0.45
DRD3 P35462 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8293216 0.94 HDAC3 (0.48) HDAC3HDAC1NPC1RAB9AHTR1A
Hydrochloric Acid SCHEMBL6809246 0.92 HDAC3 (0.47) HDAC3HDAC1NPC1RAB9AHTR1A
SCHEMBL8293671 0.88 HDAC3 (0.39) HDAC3HDAC1NPC1RAB9AHTR1A
SCHEMBL8293650 0.87 HDAC3 (0.48) HDAC3HDAC1NPC1RAB9AHTR1A
SCHEMBL8294907 0.87 HDAC3 (0.36) HDAC3HDAC1NPC1RAB9AHTR1A
SCHEMBL8294918 0.87 DRD2 (0.39) HDAC3HDAC1NPC1RAB9AHTR1A
Hydrochloric Acid SCHEMBL6805082 0.84 HDAC3 (0.46) HDAC3HDAC1NPC1RAB9AHTR1A
SCHEMBL5355999 0.83 DPP4 (0.58) HDAC3HDAC1NPC1RAB9AHTR1A
SCHEMBL8294992 0.83 DPP8 (0.41)
Hydrochloric Acid SCHEMBL5346118 0.82 DPP4 (0.57) HDAC3HDAC1NPC1RAB9AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005019168-A2 FLUORINATED LYSINE DERIVATIVES AS DIPEPTIDYL PEPTIDASE IV INHIBITORS PFIZER PRODUCTS INC. (US) 2005-03-03 WO disclosed