SCHEMBL8294709

SCHEMBL8294709

CS(=O)OCCn1c(Cl)cnc(NCCC2CCCCN2C(=O)OC(C)(C)C)c1=O

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.36
ATM Q13315 2/20 0.36
PDE8B O95263 1/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
SYK P43405 1/20 0.34
GRM5 P41594 3/20 0.33
TRPV1 Q8NER1 2/20 0.33
PRMT5 O14744 1/20 0.33
KDM1A O60341 1/20 0.33
PDE7B Q9NP56 1/20 0.33
ALDH1A1 P00352 1/20 0.33
OPRM1 P35372 1/20 0.32
OPRD1 P41143 1/20 0.32
OPRK1 P41145 1/20 0.32
OGFRL1 Q5TC84 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5475019 0.89 ATM (0.37) CHEK2ATMPDE8BALOX5APFEN1
SCHEMBL5483612 0.89 ATM (0.39) CHEK2ATMPDE8BALOX5APFEN1
SCHEMBL5479174 0.88 ATM (0.39) CHEK2ATMPDE8BALOX5APFEN1
SCHEMBL5479364 0.80 CHEK2 (0.39) CHEK2ATMPDE8BALOX5APFEN1
SCHEMBL5484745 0.80 ATM (0.39) CHEK2ATMPDE8BALOX5APFEN1
SCHEMBL5475212 0.78 ATM (0.37) CHEK2ATMPDE8BALOX5APFEN1
SCHEMBL5479053 0.77 ALDH1A1 (0.37) CHEK2IRAK4GRM5PRMT5PDE7B
SCHEMBL5483406 0.77 ALOX5AP (0.39) CHEK2ATMALOX5APFEN1IRAK4
SCHEMBL5476115 0.77 F2 (0.36) IRAK4SYKALDH1A1OPRM1OPRD1
SCHEMBL5475153 0.76 F2 (0.36) IRAK4GRM5ALDH1A1OPRM1OPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005040137-A1 AMINOALKYL-PYRAZINONES AND -PYRIDONES AS THROMBIN INHIBITORS SANTHERA PHARMACEUTICALS (SCHWEIZ) GMBH (CH) 2005-05-06 WO disclosed