SCHEMBL8294757

SCHEMBL8294757

Cc1ccc(O)c(Cn2c(NC3CCN(C)CC3)nc3ccc(C=O)cc32)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.39
NR4A2 P43354 2/20 0.39
SSTR5 P35346 5/20 0.36
SSTR4 P31391 2/20 0.36
LMNA P02545 2/20 0.36
GAA P10253 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HRH1 P35367 2/20 0.35
HRH4 Q9H3N8 2/20 0.35
SOS1 Q07889 1/20 0.35
MEN1 O00255 1/20 0.35
MLNR O43193 1/20 0.35
CACNA1F O60840 1/20 0.35
EED O75530 1/20 0.35
USP2 O75604 1/20 0.35
ABCB11 O95342 1/20 0.35
EGFR P00533 1/20 0.35
HLA-A P04439 1/20 0.35
ERBB2 P04626 1/20 0.35
TP53 P04637 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8284395 0.91 KCNH2 (0.41) KCNH2NR4A2SSTR5LMNAGAA
SCHEMBL14271789 0.91 KCNH2 (0.41) KCNH2NR4A2SSTR5LMNAGAA
SCHEMBL8293200 0.88 SSTR5 (0.53) KCNH2NR4A2SSTR5LMNAGAA
SCHEMBL8293630 0.87 KCNH2 (0.39) KCNH2NR4A2SSTR5LMNAGAA
SCHEMBL12851974 0.87 KCNH2 (0.39) KCNH2NR4A2SSTR5LMNAGAA
SCHEMBL8294929 0.87 KCNH2 (0.41) KCNH2NR4A2SSTR5LMNAGAA
SCHEMBL8294931 0.87 SSTR5 (0.37) KCNH2NR4A2SSTR5LMNAGAA
SCHEMBL8292649 0.85 KCNH2 (0.46) KCNH2NR4A2SSTR5SSTR4LMNA
SCHEMBL8294206 0.85 KCNH2 (0.43) KCNH2NR4A2SSTR5LMNAGAA
SCHEMBL8294204 0.84 KCNH2 (0.37) KCNH2NR4A2SSTR5LMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8278455-B2 5- or 6-substituted benzimidazole derivatives as inhibitors of respiratory syncytial virus replication JANSSEN PHARMACEUTICA N.V. (BE) 2012-10-02 US disclosed
US-8278455-B2 5- or 6-substituted benzimidazole derivatives as inhibitors of respiratory syncytial virus replication JANSSEN PHARMACEUTICA N.V. (BE) 2012-10-02 US disclosed
EP-1697347-B1 5- OR 6-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF RESPIRATORY SYNCYTIAL VIRUS REPLICATION TIBOTEC PHARM LTD (IE) 2011-02-23 EP disclosed
US-20090062278-A1 5- OR 6-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF RESPIRATORY SYNCYTIAL VIRUS REPLICATION JANSSEN SCIENCES IRELAND UC (IE) 2009-03-05 US disclosed
US-20090062278-A1 5- OR 6-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF RESPIRATORY SYNCYTIAL VIRUS REPLICATION JANSSEN SCIENCES IRELAND UC (IE) 2009-03-05 US disclosed
US-20070093502-A1 5- Or 6-substituted benzimidazole derivatives as inhibitors of respiratory syncytial virus replication BONFANTI JEAN-FRANCOIS 2007-04-26 US disclosed
US-20070093502-A1 5- Or 6-substituted benzimidazole derivatives as inhibitors of respiratory syncytial virus replication BONFANTI JEAN-FRANCOIS 2007-04-26 US disclosed
WO-2005058874-A1 5- OR 6-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF RESPIRATORY SYNCYTIAL VIRUS REPLICATION TIBOTEC PHARMACEUTICALS LTD. (IE) 2005-06-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070093502-A1 5- Or 6-substituted benzimidazole derivatives as inhibitors of respiratory syncytial virus replication H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, SUB1, HYOU1 KCNH2 368/4885NR4A2 331/4885SSTR5 2982/4885
US-20090062278-A1 5- OR 6-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS INHIBITORS OF RESPIRATORY SYNCYTIAL VIRUS REPLICATION H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, CYC1, SUB1 KCNH2 419/4885NR4A2 400/4885SSTR5 3585/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.