SCHEMBL8295389

SCHEMBL8295389

COc1cccc(C(=N)/C=C\N)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 1/20 0.62
PRSS2 P07478 1/20 0.62
PRSS3 P35030 1/20 0.62
PARP1 P09874 1/20 0.53
CES2 O00748 1/20 0.51
CES1 P23141 1/20 0.51
ABCG2 Q9UNQ0 1/20 0.49
NPC1 O15118 4/20 0.49
RAB9A P51151 4/20 0.49
MAOB P27338 1/20 0.47
PDE4A P27815 1/20 0.45
PDE4B Q07343 1/20 0.45
PDE4C Q08493 1/20 0.45
PDE4D Q08499 1/20 0.45
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
MAPT P10636 2/20 0.45
NFKB1 P19838 1/20 0.45
NFKB2 Q00653 1/20 0.45
RELA Q04206 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21745729 0.81 PRSS1 (0.54) PRSS1PRSS2PRSS3PARP1CES2
SCHEMBL8294719 0.79 PRSS1 (0.57) PRSS1PRSS2PRSS3PARP1CES2
SCHEMBL24454583 0.79 PRSS1 (0.65) PRSS1PRSS2PRSS3PARP1CES2
SCHEMBL23815322 0.77 PARP1 (0.48) PARP1MEN1KMT2AMAPTALDH1A1
SCHEMBL428920 0.77 PRSS1 (1.00) PRSS1PRSS2PRSS3PARP1CES2
SCHEMBL8269868 0.75 PARP1 (0.59) PRSS1PRSS2PRSS3PARP1CES2
Hydrochloric Acid SCHEMBL427173 0.75 PRSS1 (0.96) PRSS1PRSS2PRSS3PARP1CES2
Hydrochloric Acid SCHEMBL23541004 0.75 PRSS1 (0.96) PRSS1PRSS2PRSS3PARP1CES2
Hydrochloric Acid SCHEMBL28548914 0.75 PRSS1 (0.96) PRSS1PRSS2PRSS3PARP1CES2
SCHEMBL4971524 0.74 PRSS1 (0.69) PRSS1PRSS2PRSS3PARP1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005012262-A1 2-AMINOPHENYL-4-PHENYLPYRIMIDINES AS KINASE INHIBITORS CYCLACEL LIMITED (GB) 2005-02-10 WO disclosed