SCHEMBL8297150

SCHEMBL8297150

COc1ccccc1C1CCN(CCN(C(=O)C2CCCCC2)c2ccccn2)C1

nearest known ligand 0.71

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 10/20 0.71
ADRA1A P35348 6/20 0.71
DRD4 P21917 5/20 0.71
ADRA1B P35368 5/20 0.71
ADRA1D P25100 3/20 0.71
HTR7 P34969 3/20 0.71
CYP3A4 P08684 1/20 0.71
CYP2D6 P10635 1/20 0.71
TSHR P16473 1/20 0.71
HTR1B P28222 1/20 0.71
HTR2B P41595 3/20 0.70
SMN1; SMN2 Q16637 3/20 0.65
MEN1 O00255 2/20 0.65
KMT2A Q03164 2/20 0.65
LMNA P02545 2/20 0.65
BLM P54132 1/20 0.65
PMP22 Q01453 1/20 0.65
HTR2A P28223 2/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8298767 1.00 HTR1A (0.71) HTR1AADRA1ADRD4ADRA1BADRA1D
SCHEMBL8574525 1.00 HTR1A (0.71) HTR1AADRA1ADRD4ADRA1BADRA1D
SCHEMBL8296057 0.96 HTR1A (0.70) HTR1AADRA1ADRD4ADRA1BADRA1D
SCHEMBL8297779 0.95 HTR1A (0.75) HTR1AADRA1ADRD4ADRA1BADRA1D
SCHEMBL8298214 0.88 HTR1A (0.54) HTR1AADRA1ADRD4ADRA1BADRA1D
SCHEMBL8296419 0.86 HTR1A (0.63) HTR1AADRA1ADRD4ADRA1BADRA1D
SCHEMBL8300541 0.85 HTR1A (0.63) HTR1AADRA1ADRD4ADRA1BADRA1D
SCHEMBL8297225 0.85 HTR1A (0.58) HTR1AADRA1ADRD4ADRA1BADRA1D
SCHEMBL8303266 0.85 HTR1A (0.61) HTR1AADRA1ADRD4ADRA1BADRA1D
Way-100,635 SCHEMBL13398069 0.83 HTR1A (1.00) HTR1AADRA1ADRD4ADRA1BADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0898569-A1 PIPERIDINES AND PYRROLIDINES MERCK PATENT GmbH (DE) 1999-03-03 EP disclosed
WO-1997040038-A1 PIPERIDINES AND PYRROLIDINES MERCK PATENT GMBH (DE) 1997-10-30 WO disclosed