SCHEMBL8298610

SCHEMBL8298610

CC(C)(C)OC(=O)C(N)(CCc1ccc2ccccc2c1)C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC13A5 Q86YT5 1/20 0.51
CTSB P07858 1/20 0.45
CTSS P25774 1/20 0.45
CTSK P43235 1/20 0.45
CYP1A2 P05177 1/20 0.45
SLC1A3 P43003 1/20 0.41
SLC1A2 P43004 1/20 0.41
SLC1A1 P43005 1/20 0.41
HCAR2 Q8TDS4 1/20 0.40
REN P00797 2/20 0.40
PDPK1 O15530 1/20 0.40
SOX18 P35713 1/20 0.39
CHRM3 P20309 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
HIF1A Q16665 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
PPARA Q07869 1/20 0.37
CES2 O00748 1/20 0.37
PLAU P00749 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27515011 0.87 CTSB (0.47) SLC13A5CTSBCTSSCTSKCYP1A2
SCHEMBL4385270 0.85 SMN1; SMN2 (0.49) CTSBCTSSCTSKSMN1; SMN2HIF1A
SCHEMBL9544129 0.85 SMN1; SMN2 (0.49) CTSBCTSSCTSKSMN1; SMN2HIF1A
SCHEMBL9543962 0.85 SMN1; SMN2 (0.49) CTSBCTSSCTSKSMN1; SMN2HIF1A
SCHEMBL27347615 0.80 BLM (0.49) SLC13A5CTSSCTSKCYP1A2SMN1; SMN2
SCHEMBL27670635 0.80 GRM2 (0.51) SMN1; SMN2
SCHEMBL9753258 0.79 CNR2 (0.43) CTSBCTSSCTSKHDAC1HDAC8
SCHEMBL9753262 0.79 CNR2 (0.43) CTSBCTSSCTSKHDAC1HDAC8
SCHEMBL9318817 0.78 CYP1A2 (0.41) CYP1A2SMN1; SMN2
SCHEMBL8315125 0.78 SMN1; SMN2 (0.46) CTSSCTSKSMN1; SMN2HIF1AHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923550-A1 ACYLAMINOALKENYLENE-AMIDE DERIVATIVES AS NK1 AND NK2 ANTAGONISTS Novartis AG (CH) 1999-06-23 EP disclosed
WO-1998007694-A1 ACYLAMINOALKENYLENE-AMIDE DERIVATIVES AS NK1 AND NK2 ANTAGONISTS NOVARTIS AG (CH) 1998-02-26 WO disclosed