SCHEMBL8299588

SCHEMBL8299588

CC(C)(C)OC(=O)NC1CCN(c2ccc(-n3ccnc3CN3CCC3)cc2F)C1=O

nearest known ligand 0.55

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
F10 P00742 19/20 0.55
FPR2 P25090 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13958546 0.91 F10 (0.59) F10
SCHEMBL8298336 0.91 F10 (0.48) F10
SCHEMBL5691287 0.87 F10 (0.60) F10FPR2
SCHEMBL4499412 0.80 F10 (0.49) F10
SCHEMBL4513597 0.79 F10 (0.56) F10
SCHEMBL4487761 0.77 F10 (0.43) F10FPR2
SCHEMBL13958541 0.76 FPR2 (0.40) F10FPR2
SCHEMBL6365157 0.75 F10 (0.64) F10
SCHEMBL5459134 0.75 F10 (0.44) F10FPR2
SCHEMBL5710344 0.75 F10 (0.44) F10FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7482374-B2 Pyrrolidine-2-ones as Factor Xa inhibitors GLAXO GROUP LIMITED (GB) 2009-01-27 US disclosed
US-7482374-B2 Pyrrolidine-2-ones as Factor Xa inhibitors GLAXO GROUP LIMITED (GB) 2009-01-27 US disclosed
WO-2004111045-A1 PYRROLIDINE - 2- ONES AS FACTOR XA INHIBITORS GLAXO GROUP LIMITED (GB) 2004-12-23 WO disclosed