SCHEMBL8299784

SCHEMBL8299784

CC(=O)Oc1cc(Br)c(=O)[nH]n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 5/20 0.39
THRB P10828 5/20 0.39
PARP1 P09874 1/20 0.36
ALDH1A1 P00352 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
DYRK1A Q13627 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
GRIN2D O15399 1/20 0.31
GRIN3B O60391 1/20 0.31
GRIN1 Q05586 1/20 0.31
GRIN2A Q12879 1/20 0.31
GRIN2B Q13224 1/20 0.31
GRIN2C Q14957 1/20 0.31
GRIN3A Q8TCU5 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4276128 0.74 DAO (0.34) PARP1ALDH1A1KDM4EGLAGAA
SCHEMBL4420770 0.73 POLB (0.35) PARP1ALDH1A1KDM4EGLAGAA
SCHEMBL26008693 0.73 HCAR2 (0.37) THRATHRBALDH1A1DYRK1ANPC1
SCHEMBL15633292 0.69 MAPK1 (0.59) PARP1L3MBTL1GAANPC1RAB9A
SCHEMBL27725624 0.68 HPGD (0.43) ALDH1A1KDM4EGAAPDE3BPDE3A
SCHEMBL20743794 0.67
SCHEMBL30991131 0.67 HCAR2 (0.52) DAOHCAR2
SCHEMBL27906349 0.67 ALDH1A1 (0.50) ALDH1A1GAANPC1RAB9A
SCHEMBL27784137 0.67 GLA (0.40) ALDH1A1KDM4EGLAGAAGRIN2D
SCHEMBL20606968 0.66 MAP2K1 (0.37) THRATHRBKDM4ENPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004096804-A1 DIAZABICYCLONONENE AND TETRAHYDROPYRIDINE DERIVATIVES AS RENIN INHIBITORS ACTELION PHARMACEUTICALS LTD (CH) 2004-11-11 WO disclosed