SCHEMBL8301907

SCHEMBL8301907

O=C(NC(C(=O)NC1CCCCC1)c1ccccc1)c1cc(-c2ccc(OC(F)(F)F)cc2)cs1

nearest known ligand 0.73

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 9/20 0.73
MMP13 P45452 3/20 0.73
EPHX1 P07099 1/20 0.44
EPHX2 P34913 1/20 0.44
GPR88 Q9GZN0 3/20 0.43
MMP3 P08254 1/20 0.41
MMP9 P14780 1/20 0.41
MMP8 P22894 1/20 0.41
TRPV1 Q8NER1 1/20 0.41
ABL1 P00519 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TSHR P16473 2/20 0.39
USP30 Q70CQ3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6141861 0.87 MMP12 (0.64) MMP12MMP13EPHX1EPHX2MMP3
SCHEMBL6141848 0.85 MMP12 (1.00) MMP12MMP13EPHX1MMP3MMP9
SCHEMBL6141835 0.85 MMP12 (1.00) MMP12MMP13EPHX1MMP3MMP9
SCHEMBL6368500 0.85 MMP12 (1.00) MMP12MMP13EPHX1MMP3MMP9
SCHEMBL6452240 0.84 MMP12 (0.60) MMP12MMP13EPHX1EPHX2TRPV1
SCHEMBL8301905 0.80 MMP12 (0.78) MMP12MMP13EPHX2MMP3MMP9
SCHEMBL6454253 0.79 MMP12 (0.62) MMP12MMP13EPHX1EPHX2TRPV1
SCHEMBL6367993 0.77 MMP12 (0.73) MMP12MMP13EPHX1MMP3MMP9
SCHEMBL6367899 0.76 MMP12 (0.73) MMP12MMP13MMP3MMP9MMP8
SCHEMBL6530795 0.76 MMP12 (0.58) MMP12MMP13EPHX1EPHX2MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003115-A1 THIOPHENE AMINO ACID DERIVATIVES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM WARNER-LAMBERT COMPANY LLC (US) 2005-01-13 WO disclosed