SCHEMBL8302165

SCHEMBL8302165

COc1cc(CN2CCN(C(=O)CCCCC(c3ccc(F)cc3)c3ccc(F)cc3)CC2=O)cc(O)c1OC

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 14/20 0.57
CACNA1F O60840 2/20 0.41
DRD4 P21917 2/20 0.41
DRD5 P21918 2/20 0.41
HRH2 P25021 2/20 0.41
ADRA1D P25100 2/20 0.41
HTR2A P28223 2/20 0.41
HTR7 P34969 2/20 0.41
ADRA1A P35348 2/20 0.41
HRH1 P35367 2/20 0.41
ADRA1B P35368 2/20 0.41
OPRM1 P35372 2/20 0.41
DRD3 P35462 2/20 0.41
OPRD1 P41143 2/20 0.41
OPRK1 P41145 2/20 0.41
HTR6 P50406 2/20 0.41
CACNA1D Q01668 2/20 0.41
SLC6A3 Q01959 2/20 0.41
CACNA1S Q13698 2/20 0.41
CACNA1C Q13936 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5026297 0.95 KCNH2 (0.60) KCNH2CACNA1FDRD4DRD5HRH2
SCHEMBL5023972 0.86 KCNH2 (0.77) KCNH2
SCHEMBL5076819 0.81 KCNH2 (0.77) KCNH2CACNA1FDRD4DRD5HRH2
SCHEMBL5026271 0.78 KCNH2 (0.75) KCNH2SLC6A3
SCHEMBL5026247 0.75 KCNH2 (0.59) KCNH2
SCHEMBL5023632 0.73 SLC6A3 (0.48) KCNH2CACNA1FDRD4DRD5HRH2
SCHEMBL5024663 0.73 KCNH2 (0.61) KCNH2CACNA1FDRD4DRD5HRH2
SCHEMBL5024633 0.73 KCNH2 (0.79) KCNH2
SCHEMBL5076795 0.72 KCNH2 (1.00) KCNH2CACNA1FDRD4DRD5HRH2
SCHEMBL5027752 0.72 KCNH2 (0.64) KCNH2CACNA1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004089922-A2 CALCIUM CHANNEL INHIBITORS COMPRISING BENZHYDRIL SPACED FROM PIPERAZINE NEUROMED TECHNOLOGIES, INC. (CA) 2004-10-21 WO disclosed