SCHEMBL8302373

SCHEMBL8302373

NC(=O)[C@@H](N[C@@H](CC(=O)N1CCCCC1)Cc1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.48
TSHR P16473 6/20 0.43
DPP7 Q9UHL4 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C19 P33261 2/20 0.43
NPC1 O15118 1/20 0.43
CYP2D6 P10635 1/20 0.43
GAA P10253 2/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
CYP2C9 P11712 1/20 0.42
EPHX1 P07099 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306001 0.85 HPGD (0.49) HPGDTSHRTDP1CYP1A2CYP3A4
SCHEMBL8303027 0.81 EPHX1 (0.51) CYP2C19EPHX1
SCHEMBL17945538 0.75 NPC1 (0.49) HPGDTSHRDPP7TDP1CYP1A2
SCHEMBL17945842 0.73 CHRM1 (0.46) HPGDDPP7TDP1NPC1GAA
SCHEMBL26330804 0.72 HPGD (0.72) HPGDTSHRTDP1CYP1A2CYP3A4
Acetic Acid SCHEMBL6705363 0.71 DPP4 (0.62) HPGDTSHRDPP7TDP1CYP3A4
SCHEMBL7319741 0.70 NPC1 (0.51) HPGDTSHRTDP1CYP1A2CYP3A4
SCHEMBL7319738 0.70 NPC1 (0.51) HPGDTSHRTDP1NPC1GAA
SCHEMBL8305615 0.69 CNR2 (0.46) HPGDTSHRGAAKMT2AMEN1
SCHEMBL703098 0.69 HPGD (0.62) HPGDTSHRTDP1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004085661-A2 PROCESS TO CHIRAL BETA-AMINO ACID DERIVATIVES MERCK & CO., INC (US) 2004-10-07 WO disclosed