SCHEMBL8302740

SCHEMBL8302740

CN[C@H]1CC[C@@H](NC(=O)c2cc(F)cnc2OC2CCSCC2)CC1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 6/20 0.46
PDE4A P27815 1/20 0.46
PDE4D Q08499 1/20 0.46
TYK2 P29597 10/20 0.40
CNR2 P34972 2/20 0.38
CRHR1 P34998 1/20 0.38
HPGD P15428 1/20 0.37
CNR1 P21554 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303135 0.89 PDE4B (0.44) PDE4BPDE4APDE4DTYK2HPGD
SCHEMBL4187279 0.89 PDE4B (0.44) PDE4BPDE4APDE4DTYK2HPGD
Hydrochloric Acid SCHEMBL4185098 0.88 PDE4B (0.44) PDE4BPDE4APDE4DTYK2HPGD
SCHEMBL5550951 0.88 PDE4B (0.43) PDE4BPDE4APDE4DTYK2CNR2
SCHEMBL4187275 0.88 PDE4B (0.43) PDE4BPDE4APDE4DTYK2CNR2
SCHEMBL8301516 0.87 PDE4B (0.43) PDE4BPDE4APDE4DTYK2CNR2
SCHEMBL4193766 0.87 PDE4B (0.43) PDE4BPDE4APDE4DTYK2CNR2
SCHEMBL5547933 0.87 PDE4B (0.55) PDE4BPDE4APDE4DCNR2CRHR1
SCHEMBL4182884 0.86 PDE4B (0.50) PDE4BPDE4APDE4DTYK2CNR2
SCHEMBL8303245 0.86 PDE4B (0.50) PDE4BPDE4APDE4DTYK2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005009995-A1 NICOTINAMIDE DERIVATIVES USEFUL AS PDE4 INHIBITORS PFIZER LIMITED (GB) 2005-02-03 WO disclosed