SCHEMBL8303655

SCHEMBL8303655

FC(F)(F)c1ccc(CCc2cnc[nH]2)cc1

nearest known ligand 0.67

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 4/20 0.67
HRH4 Q9H3N8 3/20 0.67
CYP19A1 P11511 3/20 0.64
TAAR1 Q96RJ0 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2741585 0.81 TAAR1 (0.59) HRH3HRH4CYP19A1TAAR1
SCHEMBL6028497 0.81 HRH3 (0.68) HRH3HRH4CYP19A1TAAR1
SCHEMBL2741604 0.77 HRH4 (0.68) HRH3HRH4TAAR1
SCHEMBL224745 0.77 TAAR1 (1.00) HRH3HRH4TAAR1
SCHEMBL934227 0.75 TAAR1 (0.73) TAAR1
SCHEMBL8963903 0.75 HRH3 (0.73) HRH3HRH4TAAR1
SCHEMBL27706452 0.74 TAAR1 (0.59) TAAR1
SCHEMBL4321538 0.74 HRH3 (0.68) HRH3HRH4TAAR1
SCHEMBL7468703 0.73 HRH3 (0.73) HRH3HRH4CYP19A1TAAR1
SCHEMBL18526451 0.71 HRH3 (0.58) HRH3HRH4TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0952842-A2 A METHOD OF TREATING CANCER Merck & Co., Inc. (US) 1999-11-03 EP claimed
WO-1997038664-A2 A METHOD OF TREATING CANCER MERCK & CO., INC. (US) 1997-10-23 WO claimed