SCHEMBL8303663

SCHEMBL8303663

COC(=O)C1=C(CC(=O)N2CCN(C3CC4CCC(C3)N4C)CC2)NC(C[S+]([O-])c2ccccc2)=C(C(=O)OC)[C@H]1c1c(Cl)cccc1Cl

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.33
ALDH1A1 P00352 4/20 0.33
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
MGLL Q99685 3/20 0.32
SCD O00767 1/20 0.32
CCR3 P51677 1/20 0.32
ORAI1 Q96D31 1/20 0.31
BDKRB1 P46663 1/20 0.31
CHRM2 P08172 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
GAA P10253 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7499272 0.99 KDM4E (0.33) KDM4EALDH1A1CYP2C9CYP2C19MGLL
Hydrochloric Acid SCHEMBL8186905 0.94 KDM4E (0.32) KDM4EALDH1A1CYP2C9CYP2C19MGLL
Citric Acid SCHEMBL8188402 0.93
Hydrochloric Acid SCHEMBL8188711 0.93 KDM4E (0.32) KDM4EALDH1A1CCR3ORAI1
SCHEMBL7494164 0.93 KDM4E (0.35) KDM4EALDH1A1CYP2C9CYP2C19MGLL
Hydrochloric Acid SCHEMBL8186493 0.92 KDM4E (0.32) KDM4EALDH1A1CCR3ORAI1
Hydrochloric Acid SCHEMBL7498615 0.92 KDM4E (0.34) KDM4EALDH1A1CYP2C9CYP2C19MGLL
Hydrochloric Acid SCHEMBL8188451 0.92 DRD2 (0.35) KDM4EALDH1A1MEN1KMT2A
SCHEMBL8048899 0.89 KDM4E (0.31) KDM4EALDH1A1MEN1KMT2A
SCHEMBL8176848 0.89 KDM4E (0.31) KDM4EALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-11106375-A None JP disclosed
JP-H11106375-A OPTICALLY ACTIVE 1,4-DIHYDROPYRIDINE COMPOUND AS BRADYKININ ANTAGONIST PFIZER PHARMACEUT INC 1999-04-20 JP disclosed
EP-0899261-A1 Optical active 1,4-dihydropyridine compounds as bradykinin antagonists PFIZER INC. (US) 1999-03-03 EP disclosed