SCHEMBL8304233

SCHEMBL8304233

COc1ccc2c(n1)N(C1CC1)c1ncccc1C(=O)N2C

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.47
LMNA P02545 1/20 0.47
POLB P06746 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
MAPK1 P28482 1/20 0.47
ADORA2A P29274 1/20 0.47
ADORA1 P30542 1/20 0.47
PDE3A Q14432 1/20 0.47
MAPK7 Q13164 5/20 0.38
LRRK2 Q5S007 3/20 0.38
DCLK1 O15075 2/20 0.38
BRD4 O60885 7/20 0.35
OPRL1 P41146 2/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
BRDT Q58F21 1/20 0.33
IDH1 O75874 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8548089 0.84 ALDH1A1 (0.41) ALDH1A1LMNAPOLBADORA3MAPK1
SCHEMBL8305521 0.81 ALDH1A1 (0.47) ALDH1A1LMNAPOLBADORA3MAPK1
SCHEMBL8300415 0.80 CYP3A4 (0.45) MAPK7LRRK2DCLK1BRD4IDH1
SCHEMBL8547811 0.79 MTOR (0.42) ALDH1A1LMNAPOLBADORA3MAPK1
SCHEMBL8546272 0.79 ALDH1A1 (0.43) ALDH1A1LMNAPOLBADORA3MAPK1
SCHEMBL12427418 0.78 ALDH1A1 (0.51) ALDH1A1LMNAPOLBADORA3MAPK1
SCHEMBL8299602 0.73 ALDH1A1 (0.69) ALDH1A1LMNAPOLBADORA3MAPK1
SCHEMBL13915889 0.73 ALDH1A1 (0.63) ALDH1A1LMNAPOLBADORA3MAPK1
SCHEMBL8418964 0.70 KDM4E (0.40) ALDH1A1LMNAPOLBADORA3ADORA2A
SCHEMBL8339203 0.70 KDM4E (0.37) ALDH1A1LMNAPOLBADORA3ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0429987-B1 5,11-Dihydro-6H-dipyrido[3,2-b:2',3'-e] [1,4]diazepines and their use in the prevention or treatment of HIV infection BOEHRINGER INGELHEIM PHARMA (US) 1999-03-17 EP claimed
EP-0429987-B1 5,11-Dihydro-6H-dipyrido[3,2-b:2',3'-e] [1,4]diazepines and their use in the prevention or treatment of HIV infection BOEHRINGER INGELHEIM PHARMA (US) 1999-03-17 EP disclosed
EP-0900214-A1 PROCESS FOR PREPARATION OF PYRIMIDINE DERIVATIVES Yuhan Corporation (KR) 1999-03-10 EP disclosed
WO-1997042186-A1 PROCESS FOR PREPARATION OF PYRIMIDINE DERIVATIVES YUHAN CORPORATION (KR) 1997-11-13 WO disclosed