SCHEMBL8304601

SCHEMBL8304601

CCOC(=O)Nc1cc2ccccc2cc1Br

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.60
HPGD P15428 2/20 0.60
MAOB P27338 2/20 0.59
CYP1A2 P05177 2/20 0.54
CYP2C9 P11712 2/20 0.54
CYP2C19 P33261 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.53
F2R P25116 1/20 0.51
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
CRHBP P24387 1/20 0.49
CRHR2 Q13324 1/20 0.49
HSD17B10 Q99714 2/20 0.48
MAPT P10636 2/20 0.48
LMNA P02545 1/20 0.48
MAPK1 P28482 1/20 0.48
KDM4E B2RXH2 1/20 0.48
GLA P06280 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3827727 0.82 ALDH1A1 (0.60) ALDH1A1HPGDMAOBCYP1A2CYP2C9
SCHEMBL3829756 0.82 ALDH1A1 (0.60) ALDH1A1HPGDMAOBCYP1A2CYP2C9
SCHEMBL1188292 0.81 ALDH1A1 (0.62) ALDH1A1HPGDMAOBCYP1A2CYP2C9
SCHEMBL11642079 0.80 CYP1A2 (0.73) ALDH1A1HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL28401182 0.78 ALDH1A1 (0.72) ALDH1A1HPGDMAOBCYP1A2CYP2C9
SCHEMBL2538042 0.78 CYP1A2 (0.53) ALDH1A1HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL11656966 0.78 ALDH1A1 (0.76) ALDH1A1HPGDMAOBCYP1A2CYP2C9
SCHEMBL11765560 0.76 KDM4E (0.68) ALDH1A1HPGDMAOBCYP1A2CYP2C9
SCHEMBL11722034 0.76 CYP1A2 (0.58) ALDH1A1HPGDCYP1A2CYP2C9CYP2C19
SCHEMBL10753431 0.76 CYP1A2 (0.58) ALDH1A1HPGDCYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0650599-B1 METHOD OF COLORIMETRIC ANALYSIS OF MALONIC DIALDEHYDE AND 4-HYDROXY-2-ENALDEHYDES AS INDEXES OF LIPID PEROXIDATION, KITS FOR CARRYING OUT SAID METHOD, SUBSTITUTED INDOLES FOR USE IN SAID METHOD AND THEIR PREPARATION OXIS ISLE OF MAN LIMITED (GB) 1999-11-03 EP disclosed
US-5726063-A Method of colorimetric analysis of malonic dialdehyde and 4-hydroxy-2-enaldehydes as indexes of lipid peroxidation, kits for carrying out said method, substituted indoles for use in said method and their preparation OXIS ISLE OF MAN, LIMITED (US) 1998-03-10 US disclosed