SCHEMBL8304619

SCHEMBL8304619

Cc1ccc(-c2ccccc2CN)cc1O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 2/20 0.52
NOS3 P29474 1/20 0.51
NOS1 P29475 1/20 0.51
NOS2 P35228 1/20 0.51
APP P05067 1/20 0.44
TSHR P16473 1/20 0.40
CASP1 P29466 1/20 0.40
MCL1 Q07820 1/20 0.40
HSD17B3 P37058 1/20 0.39
PRMT5 O14744 1/20 0.38
WDR77 Q9BQA1 1/20 0.38
HTR7 P34969 1/20 0.37
PNMT P11086 1/20 0.37
F10 P00742 1/20 0.36
MAPT P10636 2/20 0.36
TRPA1 O75762 1/20 0.36
PIK3CD O00329 1/20 0.36
ABL1 P00519 1/20 0.36
EGFR P00533 1/20 0.36
HCK P08631 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27867853 0.87 DPP4 (0.52) DPP4NOS3NOS1NOS2APP
SCHEMBL9294904 0.84 DPP4 (0.57) DPP4NOS3NOS1NOS2HSD17B3
SCHEMBL3785259 0.84 DPP4 (0.57) DPP4NOS3NOS1NOS2HSD17B3
SCHEMBL5045191 0.81 DPP4 (0.57) DPP4NOS3NOS1NOS2HSD17B3
SCHEMBL1007616 0.78 MCL1 (0.59) APPTSHRCASP1MCL1HTR7
SCHEMBL27470047 0.77 APP (0.57) APPTSHRCASP1MCL1MAPT
SCHEMBL12524048 0.74 DPP4 (0.69) DPP4NOS3NOS1NOS2PNMT
SCHEMBL1038044 0.74 DPP4 (0.69) DPP4NOS3NOS1NOS2HTR7
SCHEMBL3787422 0.74 DPP4 (0.62) DPP4NOS3NOS1NOS2HTR7
SCHEMBL2450381 0.74 DPP4 (0.62) DPP4NOS3NOS1NOS2PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891333-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-01-20 EP disclosed
WO-1997036875-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO disclosed