SCHEMBL8304952

SCHEMBL8304952

CC(COc1ccc(CC2SC(=O)NC2=O)cc1)NCC(O)c1ccc2ccccc2c1

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PPARG P37231 8/20 0.59
FFAR1 O14842 11/20 0.50
PPARA Q07869 3/20 0.47
MEN1 O00255 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
KMT2A Q03164 1/20 0.46
HIF1A Q16665 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305245 0.87 PPARG (0.63) PPARGFFAR1CYP1A2CYP2D6HIF1A
SCHEMBL8406934 0.87 PPARG (0.63) PPARGFFAR1CYP1A2CYP2D6HIF1A
SCHEMBL8305440 0.87 PPARG (0.63) PPARGFFAR1CYP1A2CYP2D6HIF1A
SCHEMBL8305247 0.87 PPARG (0.63) PPARGFFAR1CYP1A2CYP2D6HIF1A
SCHEMBL8307935 0.85 PPARG (0.55) PPARGFFAR1PPARAMEN1CYP1A2
SCHEMBL8304617 0.84 PPARG (0.60) PPARGFFAR1PPARA
SCHEMBL8974677 0.83 PPARG (0.57) PPARGFFAR1PPARAMEN1CYP1A2
SCHEMBL8974649 0.81 FFAR1 (0.53) PPARGFFAR1PPARAMEN1CYP1A2
SCHEMBL8974734 0.81 FFAR1 (0.56) PPARGFFAR1PPARA
SCHEMBL8975130 0.79 FFAR1 (0.52) PPARGFFAR1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5977374-A 5-(4-hydroxy-OR 4-acetoxy-benzyl)-3- triphenylmethylthiazolidine-2,4-dione and method for producing same SANKYO COMPANY, LIMITED (JP) 1999-11-02 US disclosed
EP-0590793-B1 Oxazolidine derivatives having anti-diabetic and anti-obesity properties, their preparation and their therapeutic uses SANKYO CO (JP) 1999-10-13 EP disclosed
US-5635534-A 1-PHENYL-2-(2-PHENYLOXY OR THIO)-1-METHYLETHYL)AMINOETHANOL DERIVATIVES; ALDOSE REDUCTASE INHIBITORS; NONTOXIC; ANTIDIABETIC,-OBESITY,-LIPEMIC AND HYPOGLYCEMIC AGENTS SANKYO COMPANY, LIMITED (JP) 1997-06-03 US disclosed
US-5576340-A Aromatic amino-alcohol derivatives having anti-diabetic and anti-obesity properties, their preparation and their therapeutic uses SANKYO COMPANY, LIMITED (JP) 1996-11-19 US disclosed
EP-0543662-B1 Aromatic amino-alcohol derivatives having anti-diabetic and anti-obesity properties, their preparation and their therapeutic uses SANKYO CO (JP) 1996-09-18 EP disclosed
US-5436257-A Low toxicity SANKYO COMPANY, LIMITED (JP) 1995-07-25 US disclosed
EP-0590793-A1 Oxazolidine derivatives having anti-diabetic and anti-obesity properties, their preparation and their therapeutic uses SANKYO COMPANY LIMITED (JP) 1994-04-06 EP disclosed
EP-0543662-A2 Aromatic amino-alcohol derivatives having anti-diabetic and anti-obesity properties, their preparation and their therapeutic uses Sankyo Company Limited (JP) 1993-05-26 EP disclosed