SCHEMBL8305099

SCHEMBL8305099

O=C(c1cccs1)c1ccc(Nc2ncnc3ccc(O)cc23)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.48
RAF1 P04049 3/20 0.46
BRAF P15056 3/20 0.46
ERBB2 P04626 3/20 0.45
HPGD P15428 1/20 0.45
CASP3 P42574 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45
ALK Q9UM73 2/20 0.45
LCK P06239 1/20 0.43
RIPK2 O43353 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8308099 0.85 NPC1 (0.49) EGFRERBB2HPGDLCK
SCHEMBL8308835 0.84 HDAC3 (0.52) EGFRERBB2
SCHEMBL8307434 0.84 EGFR (0.53) EGFRRAF1BRAFERBB2ALK
Hydrochloric Acid SCHEMBL8306555 0.82 HDAC3 (0.50) EGFRERBB2
SCHEMBL7242341 0.79 EGFR (0.53) EGFRERBB2
SCHEMBL8615382 0.78 MAPK13 (0.40) BRAFHPGDCASP3SENP7SENP6
Hydrochloric Acid SCHEMBL6186793 0.75 EGFR (0.67) EGFRERBB2
SCHEMBL7240463 0.75 EGFR (0.55) EGFRBRAFERBB2
SCHEMBL7235423 0.75 EGFR (0.63) EGFRERBB2
SCHEMBL641359 0.74 EGFR (0.75) EGFRRAF1BRAFERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0790986-B1 ANILINE DERIVATIVES ZENECA LTD (GB) 1999-01-20 EP disclosed
EP-0790986-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1997-08-27 EP disclosed
WO-1996015118-A1 ANILINE DERIVATIVES ZENECA LIMITED (GB) 1996-05-23 WO disclosed