SCHEMBL8615382

SCHEMBL8615382

O=C(c1cccs1)c1ccc(Nc2ncc3cc(O)ccc3n2)cc1Cl

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK13 O15264 2/20 0.40
MAPK12 P53778 2/20 0.40
MAPK11 Q15759 2/20 0.40
MAPK14 Q16539 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
APOBEC3A P31941 1/20 0.40
APOBEC3G Q9HC16 1/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
BRAF P15056 5/20 0.38
CASP3 P42574 2/20 0.38
SENP7 Q9BQF6 2/20 0.38
SENP6 Q9GZR1 2/20 0.38
HPGD P15428 1/20 0.38
GAA P10253 2/20 0.38
ALDH1A1 P00352 1/20 0.38
MAPT P10636 1/20 0.38
AURKA O14965 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8618312 0.82 WEE1 (0.43) BRAFALDH1A1MAPT
SCHEMBL8305099 0.78 EGFR (0.48) BRAFCASP3SENP7SENP6HPGD
Hydrochloric Acid SCHEMBL8618014 0.70 BRAF (0.41) MAPK13MAPK12MAPK11MAPK14MEN1
SCHEMBL13363011 0.68 BRAF (0.55) BRAFMAPT
SCHEMBL13362984 0.67 AURKA (0.46) BRAFAURKA
SCHEMBL3429200 0.67 BRAF (0.52) MEN1KMT2ANPC1RAB9ABRAF
SCHEMBL11755917 0.67 SMN1; SMN2 (0.68) MEN1KMT2AAPOBEC3AAPOBEC3GNPC1
SCHEMBL3647900 0.66 SYK (0.46) MAP3K5
Hydrochloric Acid SCHEMBL8308099 0.66 NPC1 (0.49) MEN1KMT2ANPC1RAB9ASMN1; SMN2
SCHEMBL8308835 0.66 HDAC3 (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5821246-A USEFUL AS TYROSINE KINASE INHIBITORS AND FOR THE TREATMENT OF PROLIFERATIVE DISEASES SUCH AS CANCER ZENECA LIMITED (GB) 1998-10-13 US disclosed