SCHEMBL8305400

SCHEMBL8305400

Cc1cc(-c2ccncc2)nc2ccc3c(ncn3C)c12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPT P10636 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
LMNA P02545 1/20 0.39
RECQL P46063 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
LATS1 O95835 2/20 0.38
LATS2 Q9NRM7 1/20 0.38
HPGD P15428 1/20 0.38
GSK3B P49841 1/20 0.38
NSD3 Q9BZ95 2/20 0.36
DYRK1A Q13627 2/20 0.35
CTSS P25774 1/20 0.35
MAPK1 P28482 1/20 0.34
CYP17A1 P05093 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP11B1 P15538 1/20 0.34
PIK3CD O00329 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6825743 0.86 LATS1 (0.37) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL6822491 0.86 MAPK1 (0.41) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL6825731 0.84 LATS1 (0.38) KDM4EALDH1A1MAPTMEN1KMT2A
SCHEMBL6825653 0.74 CYP2A6 (0.45) MAPTMEN1KMT2AHPGDCTSS
SCHEMBL6825658 0.72 CYP2A6 (0.43) KMT2ALMNANPSR1LATS1LATS2
SCHEMBL6827688 0.72 CYP2A6 (0.42) MAPTMEN1KMT2ACTSSMAPK1
SCHEMBL6825775 0.69 MAP4K4 (0.40) DPP4
SCHEMBL6825776 0.68 MAP4K4 (0.39) DPP4
SCHEMBL6825733 0.67 MAP4K4 (0.46) SYK
SCHEMBL11996132 0.64 GSK3B (0.53) KDM4EALDH1A1MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004089950-A1 TRICYCLIC HETEROAROMATIC COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2004-10-21 WO disclosed