SCHEMBL8305638

SCHEMBL8305638

COCC1CN(c2ccc3nc(CO)sc3c2)C(=O)O1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.42
MAOA P21397 1/20 0.42
GRM2 Q14416 6/20 0.40
GRM5 P41594 3/20 0.40
CALML3 P27482 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3505520 0.85 GRM2 (0.39) MAOBGRM2GRM5
SCHEMBL8303678 0.84 MAPT (0.47) GRM2GRM5
SCHEMBL8310113 0.84 GRM2 (0.38) MAOBGRM2GRM5
SCHEMBL3505099 0.84 GRM2 (0.39) MAOBGRM2GRM5
SCHEMBL8305068 0.84 GRM2 (0.38) MAOBGRM2GRM5
SCHEMBL3505659 0.84 GRM2 (0.39) MAOBGRM2GRM5
SCHEMBL3504921 0.84 GRM2 (0.39) MAOBGRM2GRM5
SCHEMBL3506626 0.83 GRM2 (0.38) MAOBGRM2GRM5
SCHEMBL3503412 0.83 GRM2 (0.38) MAOBGRM2GRM5
SCHEMBL3503413 0.83 GRM2 (0.38) MAOBGRM2GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609441-B1 Oxazolidone derivatives as monoamine oxidase inhibitors EISAI CO LTD (JP) 1999-07-21 EP disclosed
US-5475014-A Monoamine oxidase inhibor; antidepressant EISAI CO., LTD. (JP) 1995-12-12 US disclosed
EP-0609441-A1 OXAZOLIDONE DERIVATIVE Eisai Co., Ltd. (JP) 1994-08-10 EP disclosed