SCHEMBL8305881

SCHEMBL8305881

Cc1ccc(CCNC(=O)c2cc(=O)[nH]c3ccc(S(=O)(=O)N4CCCC4)cc23)cc1

nearest known ligand 0.68

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.67
MAPT P10636 5/20 0.66
POLB P06746 1/20 0.66
BACE1 P56817 3/20 0.65
TP53 P04637 2/20 0.65
ALDH1A1 P00352 2/20 0.62
LMNA P02545 1/20 0.60
HTT P42858 1/20 0.60
RXFP1 Q9HBX9 1/20 0.60
TDP1 Q9NUW8 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312500 0.91 TP53 (0.78) MAPTPOLBBACE1TP53ALDH1A1
SCHEMBL8307575 0.91 BACE1 (0.65) MAPTPOLBBACE1TP53ALDH1A1
SCHEMBL8312211 0.90 MAPT (0.75) GAAMAPTPOLBBACE1TP53
SCHEMBL8312498 0.90 MAPT (0.75) GAAMAPTPOLBBACE1TP53
SCHEMBL8311209 0.90 BACE1 (0.66) MAPTPOLBBACE1TP53ALDH1A1
SCHEMBL8312029 0.90 BACE1 (0.66) MAPTPOLBBACE1TP53ALDH1A1
SCHEMBL8312221 0.90 TP53 (0.79) MAPTPOLBBACE1TP53ALDH1A1
SCHEMBL8312476 0.90 TP53 (0.79) MAPTPOLBBACE1TP53ALDH1A1
SCHEMBL8305712 0.87 MAPT (0.87) GAAMAPTPOLBBACE1TP53
SCHEMBL8304397 0.86 MAPT (0.69) MAPTPOLBBACE1TP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed