SCHEMBL8312498

SCHEMBL8312498

O=C(NCCc1ccc(Cl)cc1)c1cc(=O)[nH]c2ccc(S(=O)(=O)N3CCCCC3)cc12

nearest known ligand 0.75

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.75
POLB P06746 1/20 0.75
BACE1 P56817 3/20 0.64
TP53 P04637 1/20 0.64
KMT2A Q03164 2/20 0.61
LMNA P02545 2/20 0.60
KDM4E B2RXH2 1/20 0.60
TDP1 Q9NUW8 1/20 0.58
ALDH1A1 P00352 1/20 0.57
HTT P42858 1/20 0.57
RXFP1 Q9HBX9 1/20 0.57
GAA P10253 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312211 1.00 MAPT (0.75) MAPTPOLBBACE1TP53KMT2A
SCHEMBL8312029 0.91 BACE1 (0.66) MAPTPOLBBACE1TP53LMNA
SCHEMBL8311209 0.91 BACE1 (0.66) MAPTPOLBBACE1TP53LMNA
SCHEMBL8305881 0.90 GAA (0.67) MAPTPOLBBACE1TP53LMNA
SCHEMBL8307575 0.90 BACE1 (0.65) MAPTPOLBBACE1TP53LMNA
SCHEMBL8305790 0.90 MAPT (0.76) MAPTPOLBBACE1TP53KMT2A
SCHEMBL8304397 0.85 MAPT (0.69) MAPTPOLBBACE1TP53KMT2A
SCHEMBL8304419 0.84 MAPT (0.83) MAPTPOLBBACE1TP53KMT2A
SCHEMBL8311329 0.84 BACE1 (0.62) MAPTPOLBBACE1TP53KMT2A
SCHEMBL8312231 0.84 BACE1 (0.62) MAPTPOLBBACE1TP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed