SCHEMBL8305928

SCHEMBL8305928

Oc1cc(-c2cccnc2)cnc1Nc1ccccn1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.48
RAB9A P51151 2/20 0.48
TP53 P04637 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
EGFR P00533 3/20 0.48
L3MBTL1 Q9Y468 3/20 0.48
PDGFRB P09619 1/20 0.48
PDGFRA P16234 1/20 0.48
KDM4E B2RXH2 1/20 0.48
GRM5 P41594 1/20 0.46
CYP2A6 P11509 5/20 0.44
TSHR P16473 1/20 0.44
FGFR1 P11362 2/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALPL P05186 1/20 0.41
POLB P06746 1/20 0.41
ALPI P09923 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8310997 0.79 GRM5 (0.74) KDM4EGRM5MKNK1MKNK2ALDH1A1
SCHEMBL29517855 0.72 NPC1 (0.47) NPC1RAB9ATP53SMN1; SMN2TDP1
SCHEMBL12590014 0.70 NPC1 (0.48) NPC1RAB9ATP53SMN1; SMN2TDP1
SCHEMBL11327666 0.69 ERN1 (0.65) NPC1RAB9ATDP1EGFRL3MBTL1
SCHEMBL27241742 0.69 ALDH1A1 (0.52) NPC1RAB9ATDP1L3MBTL1KDM4E
SCHEMBL3145741 0.68 CYP2A6 (0.51) NPC1RAB9ATP53SMN1; SMN2TDP1
SCHEMBL4037525 0.68 TSHR (0.61) NPC1RAB9ATP53SMN1; SMN2TDP1
Bromide SCHEMBL11325605 0.68 ERN1 (0.63) NPC1RAB9ATDP1EGFRL3MBTL1
SCHEMBL13701560 0.68 KDR (0.81) NPC1RAB9ATP53SMN1; SMN2TDP1
SCHEMBL21296912 0.67 CYP2A6 (0.62) NPC1RAB9ATP53SMN1; SMN2EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005021529-A1 BIPYRIDYL AMINES AND ETHERS AS MODULATORS OF METABOTROPIC GLUTAMATE RECEPTOR-5 MERCK & CO., INC. (US) 2005-03-10 WO disclosed