SCHEMBL8305992

SCHEMBL8305992

CN(C1CCCCC1)S(=O)(=O)c1ccc2[nH]c(=O)cc(C(=O)NCc3ccc(F)cc3)c2c1

nearest known ligand 0.66

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 4/20 0.66
TP53 P04637 5/20 0.54
MAPT P10636 4/20 0.51
THRB P10828 1/20 0.51
BACE1 P56817 1/20 0.48
POLB P06746 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
ALDH1A1 P00352 1/20 0.46
GAA P10253 1/20 0.46
HTT P42858 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
TSHR P16473 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305720 0.92 RXFP1 (0.58) RXFP1TP53MAPTBACE1POLB
SCHEMBL8306950 0.91 KDM4E (0.57) RXFP1TP53MAPTBACE1POLB
SCHEMBL8308106 0.84 TP53 (0.58) TP53BACE1POLBMEN1KMT2A
SCHEMBL8305695 0.83 TP53 (0.65) RXFP1TP53MAPTBACE1POLB
SCHEMBL8305716 0.83 KDM4E (0.62) TP53MAPTBACE1POLBMEN1
SCHEMBL8305815 0.83 KDM4E (0.62) TP53MAPTBACE1POLBMEN1
SCHEMBL8305884 0.81 TP53 (0.49) TP53MAPTBACE1POLBMEN1
SCHEMBL8312636 0.80 TP53 (0.77) RXFP1TP53MAPTBACE1ALDH1A1
SCHEMBL8311325 0.80 TP53 (0.77) RXFP1TP53MAPTBACE1ALDH1A1
SCHEMBL8308354 0.80 KDM4E (0.51) TP53MAPTBACE1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed