SCHEMBL8306067

SCHEMBL8306067

CC(=O)N1C[C@@H](O)C[C@@H]1C(=O)N[C@H](CCCNC(=N)N)C(=O)c1nc2ccccc2s1

nearest known ligand 0.70

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PRSS1 P07477 3/20 0.70
TPSAB1 Q15661 3/20 0.70
F2 P00734 4/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4314345 1.00 PRSS1 (0.70) PRSS1TPSAB1F2
SCHEMBL5634902 1.00 PRSS1 (0.70) PRSS1TPSAB1F2
SCHEMBL4314363 1.00 PRSS1 (0.70) PRSS1TPSAB1F2
SCHEMBL5634690 1.00 PRSS1 (0.70) PRSS1TPSAB1F2
SCHEMBL20817059 1.00 PRSS1 (0.70) PRSS1TPSAB1F2
Sulfuric Acid SCHEMBL5045181 0.98 PRSS1 (0.67) PRSS1TPSAB1F2
Nitric Acid SCHEMBL5634370 0.95 PRSS1 (0.78) PRSS1TPSAB1F2
Nitric Acid SCHEMBL5634066 0.95 PRSS1 (0.78) PRSS1TPSAB1F2
Nitric Acid SCHEMBL5040734 0.95 PRSS1 (0.78) PRSS1TPSAB1F2
SCHEMBL14524837 0.91 PRSS1 (0.65) PRSS1TPSAB1F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7205384-B2 Process for preparing peptidyl heterocyclic ketone derivatives ORTHO-MCNEIL PHARMACEUTICAL INC. (US) 2007-04-17 US disclosed
US-7205384-B2 Process for preparing peptidyl heterocyclic ketone derivatives ORTHO-MCNEIL PHARMACEUTICAL INC. (US) 2007-04-17 US disclosed
WO-2005023804-A1 PEPTIDYL HETEROCYCLIC KETONE DERIVATIVES AND PREPARATION PROCESSES JANSSEN PHARMACEUTICA, N.V. (BE) 2005-03-17 WO disclosed