SCHEMBL8306090

SCHEMBL8306090

N=C(N)c1ccc(O)c(CNc2ncnc3cc(C(=O)N4CCC(O)C4)ccc23)c1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 3/20 0.40
CDK1 P06493 1/20 0.40
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
KMT2A Q03164 1/20 0.39
PDE5A O76074 2/20 0.39
HPGD P15428 1/20 0.38
THRB P10828 1/20 0.37
LOXL2 Q9Y4K0 2/20 0.36
PTK2 Q05397 4/20 0.36
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
F10 P00742 1/20 0.35
PRSS1 P07477 1/20 0.35
SUV39H1 O43463 1/20 0.35
PRMT1 Q99873 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2998619 0.88 F10 (0.46) CDK1PDE5AHPGDF10PRSS1
SCHEMBL6332101 0.87 CDK1 (0.39) VNN1CDK1RAB9ANPC1KMT2A
Hydrochloric Acid SCHEMBL6326771 0.87 F10 (0.45) CDK1PDE5AHPGDLOXL2F10
SCHEMBL6323093 0.87 F10 (0.40) CDK1KMT2APDE5AHPGDF10
Hydrochloric Acid SCHEMBL6324262 0.86 PDE5A (0.40) CDK1KMT2APDE5AHPGDF10
SCHEMBL8307162 0.84 PDE5A (0.39) CDK1PDE5AHPGDF10PRSS1
Hydrochloric Acid SCHEMBL6324175 0.83 PDE5A (0.39) CDK1PDE5AHPGDF10PRSS1
SCHEMBL6323907 0.78 CDK1 (0.50) CDK1PDE5ALOXL2SUV39H1PRMT1
Hydrochloric Acid SCHEMBL6325464 0.77 BTK (0.40) VNN1CDK1PDE5AF10PRSS1
SCHEMBL8311305 0.77 PDE5A (0.39) CDK1KMT2APDE5AHPGDSUV39H1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080970-A1 NOVEL BICYCLIC AROMATIC COMPOUNDS, THE PRODUCTION AND USE THEREOF IN THE FORM OF DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2004-09-23 WO disclosed