SCHEMBL8306225

SCHEMBL8306225

Nc1ccccc1Cn1c(Cl)nc2ccc(Br)cc2c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.45
DPP4 P27487 1/20 0.45
KMT2A Q03164 7/20 0.43
MEN1 O00255 6/20 0.43
ATM Q13315 1/20 0.43
AVPR1A P37288 1/20 0.41
ALDH1A1 P00352 4/20 0.41
HDAC1 Q13547 3/20 0.41
CYP1A2 P05177 1/20 0.41
GAA P10253 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTT P42858 1/20 0.41
KDM4E B2RXH2 2/20 0.41
MAPT P10636 2/20 0.41
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
HPGD P15428 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9952997 0.85 ALDH1A1 (0.55) KMT2AMEN1ATMAVPR1AALDH1A1
SCHEMBL3428161 0.83 DPP4 (0.61) CYP3A4DPP4KMT2AMEN1ATM
SCHEMBL8306239 0.76 DPP4 (0.71) CYP3A4DPP4
SCHEMBL8302314 0.75 DPP4 (0.79) CYP3A4DPP4
SCHEMBL31240990 0.75 CACNA2D1 (0.47) KMT2AMEN1ATMAVPR1ACYP1A2
SCHEMBL27074582 0.72 ALDH1A1 (0.46) KMT2AMEN1ALDH1A1HDAC1CYP1A2
SCHEMBL30757987 0.72 ALDH1A1 (0.46) KMT2AMEN1ALDH1A1HDAC1CYP1A2
SCHEMBL9954421 0.71 MEN1 (0.51) KMT2AMEN1ATMAVPR1AALDH1A1
SCHEMBL6797484 0.71 POLB (0.72) KMT2AMEN1ATMALDH1A1CYP1A2
SCHEMBL3425757 0.71 CYP3A4 (0.63) CYP3A4DPP4KMT2AALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004087053-A9 DIPEPTIDYL PEPTIDASE INHIBITORS SYRRX INC (US) 2004-11-11 WO disclosed
WO-2004087053-A2 DIPEPTIDYL PEPTIDASE INHIBITORS SYRRX, INC. (US) 2004-10-14 WO disclosed