SCHEMBL8306421

SCHEMBL8306421

OCC(O)CN1CC[C@@](OCc2ccccc2)(c2ccc(Cl)cc2)[C@H](OCc2ccc(F)c(F)c2F)C1

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.36
CCR3 P51677 2/20 0.36
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36
CCR1 P32246 3/20 0.34
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6098492 1.00 DRD4 (0.36) DRD4CCR3OPRM1OPRL1CCR1
SCHEMBL6098489 1.00 DRD4 (0.36) DRD4CCR3OPRM1OPRL1CCR1
SCHEMBL8312834 0.85 CCR5 (0.40) DRD4CCR3OPRM1OPRL1CCR1
SCHEMBL6096743 0.85 CCR5 (0.40) DRD4CCR3OPRM1OPRL1CCR1
SCHEMBL6096740 0.85 CCR5 (0.40) DRD4CCR3OPRM1OPRL1CCR1
SCHEMBL6274732 0.85 CCR3 (0.34) CCR3CCR1ALDH1A1
SCHEMBL6841776 0.84 BCHE (0.33) CCR3OPRM1OPRL1CCR1
SCHEMBL6095673 0.81 CCR1 (0.39) CCR1ALDH1A1
SCHEMBL6095667 0.81 CCR1 (0.39) CCR1ALDH1A1
SCHEMBL6095902 0.80 CCR1 (0.38) OPRM1CCR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004080460-A1 SUBSTITUTED PIPERIDINES AS NOVEL MDM2-p53 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2004-09-23 WO disclosed