SCHEMBL8306905

SCHEMBL8306905

CCC(C)NC(=O)c1cc(=O)[nH]c2ccc(S(=O)(=O)N3CCOCC3)cc12

nearest known ligand 0.65

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.65
ALDH1A1 P00352 3/20 0.64
PKM P14618 1/20 0.64
BACE1 P56817 3/20 0.60
GAA P10253 3/20 0.55
RXFP1 Q9HBX9 1/20 0.55
HTT P42858 1/20 0.55
KMT2A Q03164 1/20 0.54
TP53 P04637 2/20 0.53
LMNA P02545 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8308903 0.92 TP53 (0.62) KDM4EALDH1A1PKMBACE1RXFP1
SCHEMBL8312032 0.91 TP53 (0.63) KDM4EALDH1A1PKMBACE1RXFP1
SCHEMBL8312492 0.91 TP53 (0.63) KDM4EALDH1A1PKMBACE1RXFP1
SCHEMBL8308219 0.88 KDM4E (0.72) KDM4EALDH1A1PKMBACE1RXFP1
SCHEMBL8306903 0.83 KDM4E (0.74) KDM4EALDH1A1PKMBACE1GAA
SCHEMBL8311992 0.83 KDM4E (0.58) KDM4EALDH1A1PKMBACE1RXFP1
SCHEMBL8312639 0.82 TP53 (0.64) KDM4EALDH1A1PKMBACE1GAA
SCHEMBL8309383 0.81 TP53 (0.66) KDM4EALDH1A1PKMBACE1GAA
SCHEMBL8305989 0.80 MEN1 (0.68) KDM4EALDH1A1BACE1RXFP1HTT
SCHEMBL8307719 0.80 POLB (0.58) KDM4EALDH1A1PKMBACE1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed