SCHEMBL8307062

SCHEMBL8307062

CC(=NOCCOc1ccc(CC2SC(=O)N(C(c3ccccc3)(c3ccccc3)c3ccccc3)C2=O)cc1)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.55
FFAR1 O14842 8/20 0.37
HTT P42858 1/20 0.36
MAPT P10636 1/20 0.36
S1PR1 P21453 2/20 0.35
BCL2 P10415 1/20 0.35
CFTR P13569 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8307060 1.00 PPARG (0.55) PPARGFFAR1HTTMAPTS1PR1
SCHEMBL8309782 0.96 PPARG (0.51) PPARGFFAR1HTTMAPTS1PR1
SCHEMBL8309781 0.96 PPARG (0.51) PPARGFFAR1HTTMAPTS1PR1
SCHEMBL8309618 0.95 PPARG (0.50) PPARGFFAR1HTTMAPTS1PR1
SCHEMBL8309616 0.95 PPARG (0.50) PPARGFFAR1HTTMAPTS1PR1
SCHEMBL8444587 0.94 PPARG (0.51) PPARGFFAR1HTTMAPTS1PR1
SCHEMBL8304210 0.94 PPARG (0.49) PPARGFFAR1HTTMAPTS1PR1
SCHEMBL8304209 0.94 PPARG (0.49) PPARGFFAR1HTTMAPTS1PR1
SCHEMBL8305089 0.93 PPARG (0.51) PPARGFFAR1HTTMAPTS1PR1
SCHEMBL8305087 0.93 PPARG (0.51) PPARGFFAR1HTTMAPTS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5972959-A Oxime derivatives, their preparation and their therapeutic use SANKYO COMPANY, LIMITED (JP) 1999-10-26 US disclosed
EP-0753003-B1 AZIRIDINE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1999-06-16 EP disclosed
EP-0708098-B1 Oxime derivatives, their preparation and their therapeutic use SANKYO CO (JP) 1999-03-03 EP disclosed
US-5668128-A INHIBITORS OF THIOL PROTEASE, PROPHYLAXIS AND TREATMENT OF BONE DISEASES, OSTEOPOROSIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-09-16 US disclosed
EP-0708098-A1 Oxime derivatives, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1996-04-24 EP disclosed