SCHEMBL8307307

SCHEMBL8307307

[CH2]c1ccc(-c2cccc3c2OCO3)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 2/20 0.46
CHEK1 O14757 1/20 0.46
PKM P14618 1/20 0.40
TSHR P16473 1/20 0.40
ABCG2 Q9UNQ0 1/20 0.40
RIPK3 Q9Y572 1/20 0.39
DHODH Q02127 1/20 0.38
GYS1 P13807 1/20 0.38
CYP1A2 P05177 1/20 0.36
CYP1B1 Q16678 1/20 0.36
GSK3B P49841 1/20 0.35
PTPRC P08575 1/20 0.34
PTGS2 P35354 2/20 0.34
ADRA2A P08913 2/20 0.33
ADRA2B P18089 2/20 0.33
ADRA2C P18825 2/20 0.33
EED O75530 1/20 0.33
TXNRD1 Q16881 1/20 0.33
TXNRD3 Q86VQ6 1/20 0.33
TXNRD2 Q9NNW7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11390274 0.83 ABCG2 (0.50) CHEK2CHEK1PKMTSHRABCG2
SCHEMBL8309663 0.83 CHEK1 (0.41) CHEK2CHEK1PKMTSHRABCG2
SCHEMBL7594061 0.80 ABCG2 (0.55) CHEK2CHEK1PKMTSHRABCG2
SCHEMBL28643377 0.79 ALDH1A1 (0.47) CHEK2CHEK1PKMTSHRABCG2
SCHEMBL4347210 0.79 RIPK3 (0.56) CHEK2CHEK1PKMTSHRABCG2
SCHEMBL6312116 0.78 ABCG2 (0.48) CHEK2CHEK1PKMTSHRABCG2
SCHEMBL962586 0.77 CHEK1 (0.40) CHEK2CHEK1PKMTSHRABCG2
SCHEMBL22493388 0.76 CHEK2 (0.56) CHEK2CHEK1PKMTSHRDHODH
SCHEMBL1145483 0.72 ABCG2 (0.50) PKMTSHRABCG2GSK3BEED
SCHEMBL14320997 0.72 CHEK2 (0.47) CHEK2CHEK1PKMTSHRABCG2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0892795-A1 PIPERIDINYLPYRAMIDINE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1999-01-27 EP disclosed
WO-1997038992-A1 PIPERIDINYLPYRAMIDINE DERIVATIVES SUMITOMO PHARMACEUTICALS COMPANY, LIMITED (JP) 1997-10-23 WO disclosed