SCHEMBL8307633

SCHEMBL8307633

O=C(NCc1ccc2c(c1)OCO2)c1cc(=O)[nH]c2ccc(S(=O)(=O)N3CCOCC3)cc12

nearest known ligand 0.78

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.78
F2 P00734 2/20 0.78
HSD17B10 Q99714 2/20 0.78
KMT2A Q03164 3/20 0.67
LMNA P02545 3/20 0.67
HPGD P15428 3/20 0.67
MEN1 O00255 2/20 0.67
USP2 O75604 1/20 0.67
SMN1; SMN2 Q16637 1/20 0.67
KDM4E B2RXH2 4/20 0.64
TP53 P04637 1/20 0.59
TSHR P16473 1/20 0.59
BACE1 P56817 1/20 0.58
MAPT P10636 2/20 0.58
POLB P06746 1/20 0.57
PKM P14618 2/20 0.55
HTT P42858 2/20 0.55
MAPK1 P28482 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8312634 0.93 TP53 (0.68) ALDH1A1F2HSD17B10KMT2ALMNA
SCHEMBL8312202 0.92 TP53 (0.70) ALDH1A1F2HSD17B10KMT2ALMNA
SCHEMBL8308860 0.92 TP53 (0.70) ALDH1A1F2HSD17B10KMT2ALMNA
SCHEMBL8311201 0.87 HSD17B10 (0.66) ALDH1A1F2HSD17B10KMT2ALMNA
SCHEMBL8303967 0.85 TP53 (0.58) ALDH1A1F2HSD17B10KMT2ALMNA
SCHEMBL8306952 0.83 KDM4E (0.62) ALDH1A1F2HSD17B10LMNAHPGD
SCHEMBL8306903 0.80 KDM4E (0.74) ALDH1A1KMT2AHPGDMEN1KDM4E
SCHEMBL8306279 0.79 TP53 (0.75) ALDH1A1LMNAKDM4ETP53BACE1
SCHEMBL8312500 0.79 TP53 (0.78) ALDH1A1LMNAKDM4ETP53BACE1
SCHEMBL8308783 0.78 TP53 (0.75) ALDH1A1KMT2ALMNAMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004078731-A1 QUINOLINE-CARBOXYLIC ACIDS AND THE DERIVATIVES THEREOF, A FOCUSED LIBRARY 'CHEMICAL DIVERSITY RESEARCH INSTITUTE', LTD. (RU) 2004-09-16 WO disclosed