SCHEMBL8307871

SCHEMBL8307871

Fc1ccc(COCc2cccs2)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.48
POLB P06746 3/20 0.46
SLC6A3 Q01959 2/20 0.43
IDO1 P14902 2/20 0.42
AGXT P21549 2/20 0.42
DRD4 P21917 1/20 0.42
DRD5 P21918 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
LMNA P02545 2/20 0.41
TP53 P04637 1/20 0.40
RAB9A P51151 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
KCNH3 Q9ULD8 1/20 0.40
TSHR P16473 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8965090 0.85 POLB (0.46) HPGDPOLBSLC6A3IDO1AGXT
SCHEMBL4631404 0.83 TSHR (0.60) HPGDPOLBIDO1SMN1; SMN2LMNA
SCHEMBL6733610 0.82 TAAR1 (0.50) HPGDPOLBLMNARAB9AL3MBTL1
SCHEMBL7453893 0.81 TSHR (0.58) HPGDPOLBIDO1SMN1; SMN2LMNA
SCHEMBL20804374 0.81 TAAR1 (0.42) POLBLMNARAB9AL3MBTL1TSHR
SCHEMBL7453891 0.80 TSHR (0.56) HPGDPOLBSMN1; SMN2LMNARAB9A
SCHEMBL28622463 0.79 TSHR (0.60) HPGDPOLBIDO1AGXTSMN1; SMN2
SCHEMBL7989987 0.79 NPSR1 (0.46) HPGDPOLBSLC6A3NPSR1SMN1; SMN2
SCHEMBL3322765 0.78 TSHR (0.42) HPGDPOLBSMN1; SMN2LMNARAB9A
SCHEMBL3322762 0.78 TSHR (0.40) RAB9AL3MBTL1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0667855-B1 SUBSTITUTED ARYLALKYNYL- AND HETEROARYLALKYNYL-N-HYDROXYUREA INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LAB (US) 1999-03-24 EP disclosed
US-5616596-A Substituted arylalkynyl-and heteroarylalkynl-N-hydroxyurea inhibitors of leukotriene biosynthesis ABBOTT LABORATORIES (US) 1997-04-01 US disclosed
EP-0667855-A4 SUBSTITUTED ARYLALKYNYL- AND HETEROARYLALKYNYL-N-HYDROXYUREA INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS. ABBOTT LAB (US) 1996-02-21 EP disclosed
EP-0667855-A1 SUBSTITUTED ARYLALKYNYL- AND HETEROARYLALKYNYL-N-HYDROXYUREA INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LABORATORIES (US) 1995-08-23 EP disclosed
WO-1994011342-A1 SUBSTITUTED ARYLALKYNYL- AND HETEROARYLALKYNYL-N-HYDROXYUREA INHIBITORS OF LEUKOTRIENE BIOSYNTHESIS ABBOTT LABORATORIES (US) 1994-05-26 WO disclosed