SCHEMBL8308315

SCHEMBL8308315

FC(F)(F)c1cccc(CCc2ccncc2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.61
NR3C2 P08235 1/20 0.55
MIF P14174 2/20 0.51
IDO1 P14902 2/20 0.50
CHEK1 O14757 1/20 0.50
DAPK3 O43293 1/20 0.50
ROCK2 O75116 1/20 0.50
RPS6KA5 O75582 1/20 0.50
CHEK2 O96017 1/20 0.50
ABL1 P00519 1/20 0.50
PRKACA P17612 1/20 0.50
RPS6KB1 P23443 1/20 0.50
AKT1 P31749 1/20 0.50
AKT2 P31751 1/20 0.50
CLK2 P49760 1/20 0.50
GSK3A P49840 1/20 0.50
GSK3B P49841 1/20 0.50
RPS6KA3 P51812 1/20 0.50
CSNK1G2 P78368 1/20 0.50
PRKAA1 Q13131 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30063565 0.86 LTA4H (0.52) TAAR1NR3C2MIFIDO1CHEK1
SCHEMBL27706452 0.81 TAAR1 (0.59) TAAR1NR3C2MIFIDO1DAO
SCHEMBL3624339 0.79 TAAR1 (0.67) TAAR1MIFIDO1DAOHTR2A
SCHEMBL9588462 0.79 HTR2A (0.50) TAAR1NR3C2MIFIDO1CHEK1
SCHEMBL23178028 0.79 TAAR1 (0.61) TAAR1MIFIDO1DAOHTR2A
SCHEMBL17894212 0.79 TAAR1 (0.61) TAAR1NR3C2MIFIDO1DAO
SCHEMBL30777700 0.79 TAAR1 (0.61) TAAR1NR3C2MIFIDO1DAO
SCHEMBL25949968 0.79 TAAR1 (0.61) TAAR1MIFIDO1DAOHTR2A
SCHEMBL29278401 0.79 TAAR1 (0.61) TAAR1NR3C2MIFIDO1DAO
SCHEMBL11383498 0.78 TAAR1 (0.65) TAAR1MIFIDO1DAOHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0854870-A4 SUBSTITUTED IMIDAZOLES HAVING ANTI-CANCER AND CYTOKINE INHIBITORY ACTIVITY MERCK & CO INC (US) 1999-01-07 EP disclosed
EP-0854870-A1 SUBSTITUTED IMIDAZOLES HAVING ANTI-CANCER AND CYTOKINE INHIBITORY ACTIVITY Merck & Co., Inc. (US) 1998-07-29 EP disclosed
WO-1997012876-A1 SUBSTITUTED IMIDAZOLES HAVING ANTI-CANCER AND CYTOKINE INHIBITORY ACTIVITY MERCK & CO., INC. (US) 1997-04-10 WO disclosed