SCHEMBL8309216

SCHEMBL8309216

CCOc1ccc(C(C)=NO)cn1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.60
CXCR1 P25024 2/20 0.39
CXCR2 P25025 2/20 0.39
KDM4E B2RXH2 2/20 0.38
HPGD P15428 2/20 0.38
HTT P42858 2/20 0.38
NNMT P40261 1/20 0.38
ACACB O00763 5/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
LMNA P02545 1/20 0.36
GFER P55789 1/20 0.36
USP2 O75604 1/20 0.36
DGAT1 O75907 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18989339 0.82 NNMT (0.56) MAPTKDM4ENNMT
SCHEMBL29483301 0.82 NNMT (0.56) MAPTKDM4ENNMT
SCHEMBL8309518 0.82 NNMT (0.56) MAPTKDM4ENNMT
SCHEMBL22359296 0.81 MAPT (0.58) MAPTCXCR1CXCR2NNMTACACB
SCHEMBL12476476 0.80 CXCR1 (0.57) MAPTCXCR1CXCR2NNMTL3MBTL1
SCHEMBL15327912 0.80 CXCR1 (0.57) MAPTCXCR1CXCR2NNMTL3MBTL1
SCHEMBL1092552 0.79 MAPT (0.74) MAPTCXCR1CXCR2NNMTACACB
SCHEMBL8309510 0.79 MAPT (0.51) MAPTHTTACACBL3MBTL1LMNA
SCHEMBL8686473 0.79 MAPT (0.51) MAPTCXCR1CXCR2NNMTACACB
SCHEMBL8309507 0.79 MAPT (0.51) MAPTHTTACACBL3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1056840-C Oxime derivatives, their preparation and their therapeutic use SANKYO CO (JP) 2000-09-27 CN disclosed
US-5972959-A Oxime derivatives, their preparation and their therapeutic use SANKYO COMPANY, LIMITED (JP) 1999-10-26 US disclosed
EP-0708098-B1 Oxime derivatives, their preparation and their therapeutic use SANKYO CO (JP) 1999-03-03 EP disclosed
US-5780490-A A O-(2,4-OXA(OR THIA)ZOLIDINYL)PHENYLOXY(OR THIO OR AMINO) ALKYLOXIME; ALDOSE REDUCTASE INHIBITORS; ANTIDIABETIC AND -HYPOGLYCEMIC AGENTS; LIVER, SKIN AND UROGENITAL DISORDERS SANKYO COMPANY, LIMITED (JP) 1998-07-14 US disclosed
US-5703096-A ANTIDIABETIC AGENTS; ALDOSE REDUCTASE INHIBITOR SANKYO COMPANY, LIMITED (JP) 1997-12-30 US disclosed
CN-1143639-A Oxime derivatives, their preparation and their therapeutic use SANKYO CO (JP) 1997-02-26 CN disclosed
EP-0708098-A1 Oxime derivatives, their preparation and their therapeutic use SANKYO COMPANY LIMITED (JP) 1996-04-24 EP disclosed