SCHEMBL8309764

SCHEMBL8309764

N#Cc1ccc(Oc2ccc(C(c3ccccc3)(c3ccccc3)n3ccnc3)cc2)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 1/20 0.61
CYP11B2 P19099 1/20 0.61
CYP19A1 P11511 10/20 0.57
NR1I2 O75469 2/20 0.48
ADORA3 P0DMS8 2/20 0.48
TBXA2R P21731 2/20 0.48
CCKBR P32239 2/20 0.48
OPRK1 P41145 2/20 0.48
SLC6A3 Q01959 2/20 0.48
KCNH2 Q12809 2/20 0.48
NR1H4 Q96RI1 2/20 0.48
TBXAS1 P24557 2/20 0.48
CYP3A4 P08684 2/20 0.48
MEN1 O00255 1/20 0.48
SLC22A1 O15245 1/20 0.48
KCNN4 O15554 1/20 0.48
GMNN O75496 1/20 0.48
USP2 O75604 1/20 0.48
TRPM2 O94759 1/20 0.48
ABCB11 O95342 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8306981 0.85 CYP11B1 (0.61) CYP11B1CYP11B2CYP19A1NR1I2ADORA3
SCHEMBL8307152 0.83 CYP11B1 (0.67) CYP11B1CYP11B2CYP19A1NR1I2ADORA3
SCHEMBL332630 0.78 CYP11B1 (1.00) CYP11B1CYP11B2CYP19A1NR1I2ADORA3
SCHEMBL10523921 0.77 CYP19A1 (0.68) CYP11B1CYP11B2CYP19A1NR1I2ADORA3
SCHEMBL8174813 0.75 MAOB (0.40) CYP19A1MEN1LMNAMAOBOPRM1
SCHEMBL9669708 0.75 CYP11B1 (0.67) CYP11B1CYP11B2CYP19A1NR1I2ADORA3
SCHEMBL12199510 0.74 CYP11B1 (0.89) CYP11B1CYP11B2CYP19A1NR1I2ADORA3
SCHEMBL2354905 0.73 CYP19A1 (1.00) CYP11B1CYP11B2CYP19A1TBXAS1CYP3A4
SCHEMBL5320974 0.73 CYP11B1 (0.80) CYP11B1CYP11B2CYP19A1NR1I2ADORA3
SCHEMBL7156136 0.73 CYP11B1 (0.80) CYP11B1CYP11B2CYP19A1NR1I2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891333-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE Merck & Co., Inc. (US) 1999-01-20 EP disclosed
WO-1997036875-A1 INHIBITORS OF FARNESYL-PROTEIN TRANSFERASE MERCK & CO., INC. (US) 1997-10-09 WO disclosed